SCHEMBL2931914

SCHEMBL2931914

Cc1cccc(C(=O)N2C[C@H]3C[C@H]3[C@H]2CN)c1-c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 6/20 0.39
HCRTR1 O43613 5/20 0.39
APOB P04114 3/20 0.38
MTTP P55157 3/20 0.38
P2RX7 Q99572 6/20 0.37
HSD11B1 P28845 1/20 0.35
PIK3CD O00329 1/20 0.34
CYP46A1 Q9Y6A2 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2930955 0.92 HCRTR2 (0.38) HCRTR2HCRTR1APOBMTTPPIK3CD
SCHEMBL2924244 0.91 CYP46A1 (0.39) HCRTR2HCRTR1P2RX7PIK3CDCYP46A1
SCHEMBL2931040 0.91 HCRTR2 (0.40) HCRTR2HCRTR1HSD11B1PIK3CDMEN1
SCHEMBL2928151 0.90 HCRTR2 (0.35) HCRTR2HCRTR1
SCHEMBL2931912 0.86 APOB (0.38) HCRTR2HCRTR1APOBMTTPP2RX7
SCHEMBL2925493 0.85 HCRTR2 (0.37) HCRTR2HCRTR1PIK3CD
SCHEMBL2930744 0.85 HCRTR2 (0.37) HCRTR2HCRTR1PIK3CDCYP46A1
SCHEMBL2930074 0.84 SLC6A7 (0.35) HCRTR2HCRTR1
SCHEMBL2925368 0.84 HCRTR1 (0.41) HCRTR2HCRTR1
SCHEMBL2932494 0.83 HCRTR2 (0.38) HCRTR2HCRTR1CYP46A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed