SCHEMBL2930544

SCHEMBL2930544

COc1ncnc2sc(NC(=O)ON3CCC(S(=O)(=O)c4ccc(Cl)cc4)CC3)nc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.36
ADORA2A P29274 5/20 0.36
ADORA3 P0DMS8 4/20 0.36
ADORA1 P30542 2/20 0.36
GCK P35557 1/20 0.36
KCNH2 Q12809 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 2/20 0.35
USP2 O75604 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 5/20 0.35
POLB P06746 2/20 0.34
TSHR P16473 2/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
KCNQ1 P51787 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HCAR1 Q9BXC0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2932239 0.92 LMNA (0.37) GHSRADORA2AADORA3ADORA1GCK
SCHEMBL1760889 0.88 ADORA2A (0.43) GHSRADORA2AADORA3ADORA1GCK
SCHEMBL2928074 0.84 ADORA2A (0.51) ADORA2AADORA1POLBKCNQ1
SCHEMBL2930809 0.81 LMNA (0.40) ADORA2AADORA3ADORA1ALDH1A1GAA
SCHEMBL2929995 0.81 ADORA2A (0.37) ADORA2AADORA3ADORA1ALDH1A1MAPT
SCHEMBL1760902 0.80 ADORA2A (0.43) ADORA2AADORA3ADORA1GCKMAPT
SCHEMBL2929673 0.79 SCN9A (0.42) ADORA2AADORA3ADORA1
SCHEMBL2931125 0.79 EIF4E (0.41) ADORA2AADORA3ADORA1MAPT
SCHEMBL1761046 0.77 ADORA2A (0.39) ADORA2AADORA3ADORA1SMN1; SMN2ALDH1A1
SCHEMBL2930508 0.77 GPR6 (0.34) ADORA2AADORA3ADORA1SMN1; SMN2HCAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027132-B1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-09-15 EP claimed