SCHEMBL2930746

SCHEMBL2930746

COc1ncnc2sc(NC(=O)ON3CCN(Cc4cc(F)ccc4O)CC3)nc12

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.40
BCHE P06276 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ALDH1A1 P00352 1/20 0.38
GPR6 P46095 3/20 0.37
OGA O60502 1/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ADORA2A P29274 2/20 0.35
ADORA1 P30542 1/20 0.35
PIK3CA P42336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2932222 0.90 KDM4E (0.38) ALDH1A1GPR6OGAADORA2AADORA1
SCHEMBL1761031 0.89 HSD17B10 (0.43) ACHEBCHEHSD17B10ALDH1A1GPR6
SCHEMBL3050426 0.86 BCHE (0.42) ACHEBCHEGPR6OGAADORA2A
SCHEMBL2934358 0.84 ACHE (0.41) ACHEBCHEALDH1A1MAPT
SCHEMBL2930557 0.82 HTT (0.38) ALDH1A1MAPTNPSR1ADORA2AADORA1
SCHEMBL2929411 0.82 ADORA2A (0.41) ACHEALDH1A1OGAMAPTADORA2A
SCHEMBL2931169 0.82 OGA (0.38) ACHEGPR6OGAADORA2AADORA1
SCHEMBL2930809 0.81 LMNA (0.40) ACHEALDH1A1MAPTADORA2AADORA1
SCHEMBL2930506 0.81 GPR6 (0.38) ACHEALDH1A1GPR6
SCHEMBL2932276 0.81 CYP2D6 (0.41) ALDH1A1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027132-B1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-09-15 EP claimed