SCHEMBL3050426

SCHEMBL3050426

COc1ncnc2sc(NC(=O)ON3CCN(Cc4cccc(F)c4O)CC3)nc12

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.42
ACHE P22303 4/20 0.42
GPR6 P46095 3/20 0.37
ADORA3 P0DMS8 2/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
LPAR2 Q9HBW0 2/20 0.34
TSHR P16473 1/20 0.34
RORC P51449 1/20 0.33
DHODH Q02127 1/20 0.33
OGA O60502 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2934358 0.91 ACHE (0.41) BCHEACHERORCDHODHHTT
SCHEMBL1760988 0.88 BCHE (0.43) BCHEACHEGPR6ADORA3ADORA2A
SCHEMBL2930746 0.86 ACHE (0.40) BCHEACHEGPR6ADORA2AADORA1
SCHEMBL2929411 0.85 ADORA2A (0.41) ACHEADORA3ADORA2AADORA1MEN1
SCHEMBL2932222 0.85 KDM4E (0.38) GPR6ADORA3ADORA2AADORA1MEN1
SCHEMBL2931169 0.84 OGA (0.38) ACHEGPR6ADORA2AADORA1MEN1
SCHEMBL3049811 0.84 MEN1 (0.42) ACHEADORA2AMEN1KMT2ALPAR2
SCHEMBL2930557 0.83 HTT (0.38) ADORA3ADORA2AADORA1MEN1KMT2A
SCHEMBL2930504 0.83 FAAH (0.45) GPR6MEN1KMT2ATSHRHTT
SCHEMBL2930809 0.82 LMNA (0.40) ACHEADORA3ADORA2AADORA1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027132-B1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-09-15 EP claimed