SCHEMBL2932222

SCHEMBL2932222

COc1ncnc2sc(NC(=O)ON3CCN(Cc4cc(Cl)ccc4O)CC3)nc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 2/20 0.36
MEN1 O00255 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 2/20 0.36
ERCC1 P07992 2/20 0.36
ERCC4 Q92889 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CASP1 P29466 1/20 0.36
CYP2C19 P33261 1/20 0.36
CASP7 P55210 1/20 0.36
GPR6 P46095 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2930746 0.90 ACHE (0.40) ALDH1A1GPR6OGAADORA2AADORA1
SCHEMBL2930557 0.89 HTT (0.38) ALDH1A1MEN1KMT2ASMN1; SMN2RAB9A
SCHEMBL1761069 0.89 FAAH (0.42) KDM4EALDH1A1TSHRMEN1ALOX15
SCHEMBL2930809 0.88 LMNA (0.40) KDM4EALDH1A1MEN1MAPK1KMT2A
SCHEMBL2930497 0.88 GPR6 (0.35) KDM4ESMN1; SMN2GPR6EPHX2ADORA3
SCHEMBL3049811 0.86 MEN1 (0.42) ALDH1A1TSHRMEN1MAPK1KMT2A
SCHEMBL2930508 0.86 GPR6 (0.34) SMN1; SMN2GPR6ADORA3ADORA2AADORA1
SCHEMBL3050426 0.85 BCHE (0.42) TSHRMEN1KMT2ASMN1; SMN2GPR6
SCHEMBL2929411 0.84 ADORA2A (0.41) KDM4EALDH1A1TSHRMEN1MAPK1
SCHEMBL2934358 0.84 ACHE (0.41) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027132-B1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-09-15 EP claimed