SCHEMBL2931358

SCHEMBL2931358

COc1ncnc2sc(NC(=O)ON3CCN(CCc4ccccc4)CC3)nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.40
AURKA O14965 1/20 0.40
GAA P10253 2/20 0.40
TSHR P16473 1/20 0.40
POLB P06746 1/20 0.39
ABCC1 P33527 1/20 0.39
MAPK1 P28482 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
ADORA2A P29274 2/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA1 P30542 1/20 0.38
LMNA P02545 1/20 0.37
HTR1A P08908 2/20 0.37
HTR1D P28221 2/20 0.37
HTR1B P28222 2/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR7 P34969 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2929411 0.91 ADORA2A (0.41) GAATSHRMAPK1ALDH1A1MAPT
SCHEMBL1761051 0.88 MAPK1 (0.48) NPSR1AURKAGAATSHRPOLB
SCHEMBL2931169 0.84 OGA (0.38) ADORA2AADORA1LMNA
Trifluoroacetic Acid SCHEMBL1761052 0.84 ACHE (0.46) NPSR1AURKAGAATSHRPOLB
SCHEMBL2930809 0.83 LMNA (0.40) GAAMAPK1ALDH1A1MAPTADORA2A
SCHEMBL3049811 0.83 MEN1 (0.42) TSHRMAPK1ALDH1A1MAPTADORA2A
SCHEMBL2930506 0.81 GPR6 (0.38) ALDH1A1LMNA
SCHEMBL2931204 0.81 GPR6 (0.47)
SCHEMBL2927982 0.81 ADORA2B (0.47) GAAALDH1A1ADORA2AADORA1SIGMAR1
SCHEMBL2931875 0.81 ALDH1A1 (0.40) GAAALDH1A1MAPTADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027132-B1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-09-15 EP claimed