SCHEMBL29314122

SCHEMBL29314122

CCN(C(=O)Cc1c(-n2cc[nH]c2=O)cc(C(F)(F)F)cc1C(F)(F)F)c1ccc(F)c(Cl)n1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 1/20 0.34
GAA P10253 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
POLQ O75417 6/20 0.33
MCOLN3 Q8TDD5 1/20 0.33
CCNE1 P24864 1/20 0.32
GRK2 P25098 1/20 0.32
CDK3 Q00526 1/20 0.32
XPO1 O14980 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CMA1 P23946 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29314119 0.91 CRHR1 (0.36) CRHR1GAANPSR1POLQMEN1
SCHEMBL29314118 0.83 POLQ (0.33) GAAPOLQMCOLN3CCNE1GRK2
SCHEMBL29314123 0.82 ALDH1A1 (0.34) CRHR1GAANPSR1POLQALDH1A1
SCHEMBL29314114 0.75 POLQ (0.32) GAAPOLQMCOLN3ALDH1A1POLB
SCHEMBL29314117 0.74 POLQ (0.31) POLQ
SCHEMBL29313854 0.69 POLB (0.31) POLB
SCHEMBL29314307 0.67 GAA (0.32) GAAPOLQ
SCHEMBL29314469 0.65 CRHR1 (0.38) CRHR1NPSR1CCNE1GRK2CDK3
SCHEMBL31009122 0.63 POLQ (0.36) CRHR1POLQ
SCHEMBL29314125 0.63 SMN1; SMN2 (0.40) GAANPSR1POLQKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed