SCHEMBL29314127

SCHEMBL29314127

CCN(C(=O)Cc1c(C(=N)/N=C\N)cc(C(F)(F)F)cc1C(F)(F)F)c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLQ O75417 15/20 0.41
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 2/20 0.35
GAA P10253 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29314165 0.83 GAA (0.33) POLQNPSR1GAAKDM4EALDH1A1
SCHEMBL29314130 0.83 RORC (0.34) POLQNPSR1GAAKDM4EALDH1A1
SCHEMBL29314172 0.83 POLQ (0.36) POLQNPSR1GAAKDM4EALDH1A1
SCHEMBL29314121 0.70 POLQ (0.44) POLQSMN1; SMN2NPSR1GAAKDM4E
SCHEMBL29314181 0.70 GAA (0.33) POLQNPSR1GAA
SCHEMBL29314183 0.70 GAA (0.30) NPSR1GAA
SCHEMBL29314167 0.69 POLQ (0.37) POLQNPSR1GAAKDM4EALDH1A1
SCHEMBL21785057 0.61 OPRM1 (0.49) SMN1; SMN2GAAKDM4EALDH1A1POLB
SCHEMBL24795106 0.61 MLYCD (0.49) SMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL8443789 0.60 SMN1; SMN2 (0.47) SMN1; SMN2NPSR1GAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed