SCHEMBL29314121

SCHEMBL29314121

CCN(C(=O)Cc1c(-c2cn[nH]c2)cc(C(F)(F)F)cc1C(F)(F)F)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLQ O75417 13/20 0.44
NPSR1 Q6W5P4 2/20 0.39
GAA P10253 1/20 0.39
ROCK2 O75116 2/20 0.38
ROCK1 Q13464 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RET P07949 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29315913 0.78 ROCK1 (0.39) ROCK2ROCK1
SCHEMBL29315909 0.77 ROCK2 (0.46) ROCK2ROCK1
SCHEMBL31009157 0.72 POLQ (0.46) POLQROCK2ROCK1
SCHEMBL29314127 0.70 POLQ (0.41) POLQNPSR1GAASMN1; SMN2KDM4E
SCHEMBL29314126 0.70 ROCK2 (0.34) ROCK2ROCK1
SCHEMBL31009207 0.67 POLQ (0.50) POLQROCK2
SCHEMBL29316278 0.66 NPBWR1 (0.39) ROCK2ROCK1
SCHEMBL29314124 0.64 SMN1; SMN2 (0.40) POLQNPSR1GAASMN1; SMN2KDM4E
SCHEMBL30716959 0.61 POLQ (0.70) POLQ
SCHEMBL29135502 0.61 POLQ (0.70) POLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed