SCHEMBL2932978

SCHEMBL2932978

O=S(O)c1ccccc1F.[Na]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.39
CES1 P23141 3/20 0.39
G6PD P11413 1/20 0.39
ALDH1A1 P00352 2/20 0.37
ALOX15 P16050 1/20 0.37
NPC1 O15118 2/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
KCNH2 Q12809 1/20 0.34
ACHE P22303 1/20 0.33
GAA P10253 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
BCHE P06276 1/20 0.32
NFE2L2 Q16236 1/20 0.32
HPGD P15428 2/20 0.32
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5354555 0.98 CES2 (0.41) CES2CES1G6PDALDH1A1ALOX15
SCHEMBL2932974 0.95 CES2 (0.39) CES2CES1G6PDALDH1A1ALOX15
SCHEMBL5042526 0.79 CES2 (0.45) CES2CES1G6PDALDH1A1ALOX15
SCHEMBL9153083 0.79 G6PD (0.50) CES2CES1G6PDALDH1A1ALOX15
SCHEMBL11859134 0.76 G6PD (0.48) CES2CES1G6PDALDH1A1ALOX15
SCHEMBL31236603 0.76 CES2 (0.37) CES2CES1G6PDALDH1A1ALOX15
SCHEMBL11423428 0.74 CES2 (0.35) CES2CES1G6PDALDH1A1NPC1
SCHEMBL29463779 0.73 CYP3A4 (0.43) G6PDALDH1A1ALOX15NPC1RAB9A
SCHEMBL9152680 0.73 CYP3A4 (0.43) G6PDALDH1A1ALOX15NPC1RAB9A
SCHEMBL9151925 0.72 G6PD (0.44) CES2CES1G6PDALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796380-A 2-allyl-3-sulfonyl-3-butenoate compound and preparation method thereof 南京工业大学 2019-05-24 CN disclosed
CN-105906537-A One-pot synthesis method of (Z)-type sulfonyl olefine acid ester compound 湖南科技学院 2016-08-31 CN disclosed
EP-2229358-A1 INDOLES AND THEIR THERAPEUTIC USE Pulmagen Therapeutics (Asthma) Limited (GB) 2010-09-22 EP disclosed
CN-101801962-A Trisubstituted pyrimidine derivatives for the treatment of proliferative diseases ASTRAZENECA AB 2010-08-11 CN disclosed
EP-2074118-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES AstraZeneca AB (SE) 2009-07-01 EP disclosed
WO-2009077728-A1 INDOLES AND THEIR THERAPEUTIC USE ARGENTA DISCOVERY LIMITED (GB) 2009-06-25 WO disclosed
US-20090018134-A1 Compounds - 945 ASTRAZENECA AB (SE) 2009-01-15 US disclosed
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed
CN-1902168-A Novel 1, 3-disubstituted azetidine derivatives as 5-HT 2A receptor ligands MERCK SHARP & DOHME (GB) 2007-01-24 CN disclosed
US-7094777-B2 5-HT2A receptor ligands MERK SHARP & DOHME LTD. 2006-08-22 US disclosed
US-20050101586-A1 Novel 5-HT2A receptor ligands MERCK SHARP & DOHME LTD. (GB) 2005-05-12 US disclosed
CN-1373112-A Method for producing allyl halide SUMITOMO CHEMICAL CO (JP) 2002-10-09 CN disclosed
EP-1231197-A1 Process for producing allyl halide compound SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-08-14 EP disclosed
US-20020107422-A1 Process for producing allyl halide compound SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2002-08-08 US disclosed
US-5100460-A HERBICIDAL COMPOUNDS AND COMPOSITIONS CONTAINING THEM RHONE-POULENC AGROCHIMIE (FR) 1992-03-31 US disclosed
CN-1039805-A Herbicidal compound and composition thereof RHONE POULENC AGROCHIMIE (FR) 1990-02-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050101586-A1 Novel 5-HT2A receptor ligands HTR2A, HTR1A, HTR5A CES2 1068/4885CES1 1984/4885G6PD 2985/4885
US-20090018134-A1 Compounds - 945 MTOR, PIK3CA, PIK3R5 CES2 2150/4885CES1 2220/4885G6PD 550/4885
US-20020107422-A1 Process for producing allyl halide compound ENY2, ZYX, RPS4Y1 CES2 1967/4885CES1 1097/4885G6PD 3142/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.