SCHEMBL2940289

SCHEMBL2940289

CS(=O)(=O)c1ccc(N2CCC(C(N)=S)C2)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 13/20 0.47
NOTUM Q6P988 1/20 0.42
AOC3 Q16853 2/20 0.41
KCNH2 Q12809 2/20 0.40
GPR55 Q9Y2T6 1/20 0.40
GPR119 Q8TDV5 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2940287 1.00 SLC6A9 (0.47) SLC6A9NOTUMAOC3KCNH2GPR55
SCHEMBL2937599 0.89 SLC6A9 (0.50) SLC6A9NOTUMAOC3KCNH2GPR55
SCHEMBL2937602 0.89 SLC6A9 (0.50) SLC6A9NOTUMAOC3KCNH2GPR55
SCHEMBL2939303 0.85 NOTUM (0.60) SLC6A9NOTUM
SCHEMBL2939305 0.85 NOTUM (0.60) SLC6A9NOTUM
SCHEMBL13363551 0.81 SLC6A9 (0.50) SLC6A9NOTUMAOC3KCNH2GPR119
SCHEMBL2937750 0.81 SLC6A9 (0.51) SLC6A9KCNH2GPR55GPR119
SCHEMBL2937751 0.81 SLC6A9 (0.51) SLC6A9KCNH2GPR55GPR119
SCHEMBL2184348 0.78 SLC6A9 (0.56) SLC6A9AOC3KCNH2GPR55GPR119
SCHEMBL2939585 0.77 SLC6A9 (0.48) SLC6A9NOTUMKCNH2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134704-B1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF GPR119 ACTIVITY IRM LLC (BM) 2010-09-22 EP disclosed
US-20100120807-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF GPR119 ACTIVITY IRM LLC (BM) 2010-05-13 US disclosed
EP-2134704-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF GPR119 ACTIVITY IRM LLC (BM) 2009-12-23 EP disclosed
WO-2008109702-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF GPR119 ACTIVITY IRM LLC (BM) 2008-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100120807-A1 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF GPR119 ACTIVITY GPR119, GPR65, GPR39 SLC6A9 2063/4885NOTUM 4356/4885AOC3 3304/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.