SCHEMBL29439722

SCHEMBL29439722

COC(=O)c1cccc(C(F)(F)F)c1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 6/20 0.51
ALDH1A1 P00352 2/20 0.51
HSD17B10 Q99714 1/20 0.51
LMNA P02545 2/20 0.45
GAA P10253 2/20 0.45
TSHR P16473 1/20 0.44
PTGS1 P23219 1/20 0.44
PDK2 Q15119 2/20 0.43
NOTUM Q6P988 1/20 0.43
RBP4 P02753 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA5A P35218 1/20 0.42
CA9 Q16790 1/20 0.42
TAS2R14 Q9NYV8 1/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
ATM Q13315 1/20 0.42
PDK1 Q15118 1/20 0.42
PDK3 Q15120 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3531721 1.00 CFTR (0.51) CFTRALDH1A1HSD17B10LMNAGAA
SCHEMBL2085863 0.85 CFTR (0.55) CFTRALDH1A1HSD17B10GAATSHR
SCHEMBL9120474 0.84 CFTR (0.46) CFTRALDH1A1HSD17B10LMNAGAA
SCHEMBL7322634 0.83 PTGS1 (0.55) CFTRHSD17B10LMNAGAATSHR
SCHEMBL11696222 0.83 HSD17B10 (0.55) ALDH1A1HSD17B10GAATSHRPDK2
SCHEMBL45490 0.82 LMNA (0.59) CFTRALDH1A1HSD17B10LMNAGAA
SCHEMBL2895994 0.82 ALDH1A1 (0.67) CFTRALDH1A1HSD17B10LMNAGAA
SCHEMBL726068 0.81 TAS2R14 (0.54) CFTRALDH1A1HSD17B10LMNAGAA
SCHEMBL5239843 0.81 CTSS (0.51) CFTRALDH1A1HSD17B10LMNAGAA
SCHEMBL1508457 0.81 LMNA (0.50) CFTRALDH1A1HSD17B10LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed