SCHEMBL29439832

SCHEMBL29439832

Cc1nccc(CO)c1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
LMNA P02545 3/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
ALOX12 P18054 1/20 0.39
NOS3 P29474 4/20 0.39
NOS2 P35228 4/20 0.39
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 1/20 0.37
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
PDXK O00764 1/20 0.37
AOX1 Q06278 1/20 0.37
CYP2A6 P11509 1/20 0.36
TRIM24 O15164 1/20 0.36
TRIM33 Q9UPN9 1/20 0.36
CYP19A1 P11511 1/20 0.35
MAOA P21397 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28714994 1.00 KDM4E (0.39) KDM4ELMNATP53MAPTTSHR
SCHEMBL26489048 0.81 NOS2 (0.44) KDM4EMAPTNOS3NOS2MEN1
SCHEMBL4795960 0.78 KDM4E (0.41) KDM4ELMNATP53MAPTTSHR
SCHEMBL29259211 0.77 GABRP (0.46) KDM4ELMNAMAPTNOS3NOS2
SCHEMBL3679899 0.77 KDM4E (0.47) KDM4ELMNATP53MAPTTSHR
SCHEMBL2355840 0.77 KDM4E (0.52) KDM4ELMNATP53MAPTTSHR
SCHEMBL30073071 0.76 NOS3 (0.36) KDM4ENOS3NOS2HPGDHSD17B10
SCHEMBL23012667 0.75 NOS2 (0.54) KDM4ELMNATP53MAPTTSHR
Hydrochloric Acid SCHEMBL28811005 0.75 TRIM24 (0.51) KDM4ELMNATP53MAPTTSHR
SCHEMBL3940135 0.75 RECQL (0.39) KDM4ELMNATP53MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3976597-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE Janssen Pharmaceutica NV (BE) 2022-04-06 EP disclosed