Dimethindene

Dimethindene

SCHEMBL29455130

C[C@@H](C1=C(CCN(C)C)Cc2ccccc21)c1ccccn1.O=C(O)/C=C\C(=O)O

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Dimethindene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 8/20 0.82
CHRM1 P11229 20/20 0.82
CHRM2 P08172 19/20 0.82
CHRM4 P08173 19/20 0.82
CHRM5 P08912 19/20 0.82
CHRM3 P20309 19/20 0.82
CYP2D6 P10635 3/20 0.82
KCNH2 Q12809 3/20 0.82
CYP1A2 P05177 1/20 0.82
CYP2C9 P11712 1/20 0.82
TSHR P16473 1/20 0.82
CYP2C19 P33261 1/20 0.82
HTR1A P08908 1/20 0.82
ADRA2A P08913 1/20 0.82
DRD1 P21728 1/20 0.82
PTGS1 P23219 1/20 0.82
SLC6A2 P23975 1/20 0.82
SLC6A4 P31645 1/20 0.82
ADRA1A P35348 1/20 0.82
OPRM1 P35372 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethindene SCHEMBL29887834 1.00 CHRM1 (0.82) CHRM1CHRM2CHRM4CHRM5CHRM3
Dimethindene SCHEMBL1972832 1.00 CHRM1 (0.82) CHRM1CHRM2CHRM4CHRM5CHRM3
Dimethindene SCHEMBL359490 1.00 CHRM1 (0.82) CHRM1CHRM2CHRM4CHRM5CHRM3
Dimethindene SCHEMBL19284560 0.90 CHRM1 (1.00) CHRM1CHRM2CHRM4CHRM5CHRM3
Dimethindene SCHEMBL30436315 0.90 CHRM1 (1.00) CHRM1CHRM2CHRM4CHRM5CHRM3
(S)-(+)-Dimethindene SCHEMBL30910954 0.90 CHRM1 (1.00) CHRM1CHRM2CHRM4CHRM5CHRM3
Dimethindene SCHEMBL29676184 0.90 CHRM1 (1.00) CHRM1CHRM2CHRM4CHRM5CHRM3
Dimethindene SCHEMBL18759 0.90 CHRM1 (1.00) CHRM1CHRM2CHRM4CHRM5CHRM3
Dimethindene SCHEMBL28142887 0.81 CHRM1 (0.76) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL6276908 0.78 HRH1 (1.00) CHRM1CHRM2CHRM4CHRM5CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119979473-A Method for forming bovine primordial germ cell-like cells by differentiating bovine iPSCs 内蒙古大学 2025-05-13 CN claimed
CN-118345027-B 3D suspension culture method capable of maintaining characteristics of expanded pluripotent stem cells 深圳市北科源细胞科技有限公司 2025-03-25 CN claimed
CN-119193473-A Method for obtaining expansile pluripotent stem cells from peripheral blood mononuclear cells by reprogramming 深圳市北科源细胞科技有限公司 2024-12-27 CN claimed
CN-118345027-A 3D suspension culture method capable of maintaining characteristics of expanded pluripotent stem cells 深圳市北科源细胞科技有限公司 2024-07-16 CN claimed
EP-3334820-B1 INDUCED EXTENDED PLURIPOTENT STEM CELLS, METHODS OF MAKING AND USING BEIHAO STEM CELL AND REGENERATIVE MEDICINE RES INSTITUTE CO LTD (CN) 2024-05-15 EP claimed
CN-117736974-A Application of DAPT in maintaining multipotency of expanded multipotential stem cells and improving proliferation capacity of multipotential stem cells 呈诺再生医学科技(北京)有限公司 2024-03-22 CN claimed
CN-116355837-A EPSC suspension culture and neural stem cell differentiation method 呈诺再生医学科技(北京)有限公司 2023-06-30 CN claimed
US-20260132373-A1 BOVINE BLASTOCYST LIKE STRUCTURES AND USES THEREOF BOARD OF SUPERVISORS OF LOUISIANA STATE UNIV AND AGRICULTURAL AND MECHANICAL COLLEGE (US) 2026-05-14 US disclosed
US-12467917-B2 Reconstructing human early embryogenesis in vitro with pluripotent stem cells CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2025-11-11 US disclosed
EP-4569013-A1 BOVINE BLASTOCYST LIKE STRUCTURES AND USES THEREOF Board of Supervisors of Louisiana State University and Agricultural and Mechanical College (US) 2025-06-18 EP disclosed
US-20250188422-A1 INDUCED TOTIPOTENT POTENTIAL STEM CELLS, METHODS OF MAKING AND USING PEKING UNIVERSITY (CN) 2025-06-12 US disclosed
CN-119979473-A Method for forming bovine primordial germ cell-like cells by differentiating bovine iPSCs 内蒙古大学 2025-05-13 CN disclosed
CN-119913110-A Method for producing high-proportion chimeric living monkey by utilizing embryonic stem cells 中国科学院脑科学与智能技术卓越创新中心 2025-05-02 CN disclosed
US-20230073534-A1 MODULATING TLR/NF-KB AND P53 SIGNALING PATHWAYS TO ENHANCE INTERSPECIES CHIMERISM BETWEEN EVOLUTIONARYILY DISTANT SPECIES THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-03-09 US disclosed
US-20220389376-A1 Methods for Reprogramming Cells NANTES UNIVERSITE (FR) 2022-12-08 US disclosed
WO-2022242455-A1 METHOD FOR INDUCING DIFFERENTIATION OF EXTENDED PLURIPOTENT STEM CELLS INTO CARDIOMYOCYTES AND APPLICATION THEREOF 湖北大学 2022-11-24 WO disclosed
US-20220308041-A1 RECONSTRUCTING HUMAN EARLY EMBRYOGENESIS IN VITRO WITH PLURIPOTENT STEM CELLS CALIFORNIA INSTITUTE OF TECHNOLOGY 2022-09-29 US disclosed
EP-4058565-A1 METHODS FOR REPROGRAMMING CELLS Monash University (AU) 2022-09-21 EP disclosed
US-20220177862-A1 Precise Gene Activation Via Novel Designed Proteins Mediating Epigenetic Remodeling NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-06-09 US disclosed
US-20220090023-A1 METHODS FOR REGULATING POTENCY OF PLURIPOTENT STEM CELLS AND APPLICATIONS THEREOF ACADEMIA SINICA (TW) 2022-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260132373-A1 BOVINE BLASTOCYST LIKE STRUCTURES AND USES THEREOF STAT3, SMAD2, LIFR HRH1 1967/4885CHRM1 4553/4885CHRM2 4290/4885
US-20220090023-A1 METHODS FOR REGULATING POTENCY OF PLURIPOTENT STEM CELLS AND APPLICATIONS THEREOF CDYL, ZFX, CDYL2 HRH1 4766/4885CHRM1 4776/4885CHRM2 4788/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.