Tilbroquinol

Tilbroquinol

SCHEMBL29465197

Cc1cc(Br)c(O)c2ncccc12

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.72
HTT P42858 7/20 0.72
HSP90AA1 P07900 7/20 0.72
TP53 P04637 6/20 0.72
SMN1; SMN2 Q16637 6/20 0.72
MEN1 O00255 5/20 0.72
KMT2A Q03164 5/20 0.72
TDP1 Q9NUW8 5/20 0.72
USP2 O75604 3/20 0.72
COMT P21964 2/20 0.57
SLC6A2 P23975 4/20 0.54
CCR1 P32246 2/20 0.54
CCR8 P51685 2/20 0.54
LMNA P02545 5/20 0.49
ALDH1A1 P00352 5/20 0.49
ALOX15 P16050 4/20 0.49
MAPT P10636 4/20 0.49
MMP14 P50281 3/20 0.49
ALOX12 P18054 3/20 0.49
MAPK1 P28482 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tilbroquinol SCHEMBL1441958 1.00 KDM4E (0.72) KDM4EHTTHSP90AA1TP53SMN1; SMN2
SCHEMBL13283110 0.86 HSP90AA1 (0.72) KDM4EHTTHSP90AA1TP53SMN1; SMN2
Broxyquinoline SCHEMBL115293 0.84 KDM4E (1.00) KDM4EHTTHSP90AA1TP53SMN1; SMN2
SCHEMBL318630 0.84 HTT (0.59) KDM4EHTTHSP90AA1TP53SMN1; SMN2
SCHEMBL29577465 0.84 HTT (0.59) KDM4EHTTHSP90AA1TP53SMN1; SMN2
SCHEMBL17046868 0.84 HTT (0.59) KDM4EHTTHSP90AA1TP53SMN1; SMN2
Broxyquinoline SCHEMBL30485535 0.84 KDM4E (1.00) KDM4EHTTHSP90AA1TP53SMN1; SMN2
Broxyquinoline SCHEMBL29607319 0.84 KDM4E (1.00) KDM4EHTTHSP90AA1TP53SMN1; SMN2
Broxyquinoline SCHEMBL31157810 0.82 KDM4E (0.96) KDM4EHTTHSP90AA1TP53SMN1; SMN2
Broxyquinoline SCHEMBL22734870 0.82 KDM4E (0.96) KDM4EHTTHSP90AA1TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250367232-A1 HALOGEN TREATMENT OF HEART ATTACK AND ISCHEMIC INJURY HUTCHINSON FRED CANCER RES (US) 2025-12-04 US disclosed
US-12203124-B2 Methods for improved rapid antimicrobial susceptibility testing SeLux Diagnostics, Inc. (US) 2025-01-21 US disclosed
US-12016880-B2 Halogen treatment of heart attack and ischemic injury FRED HUTCHINSON CANCER CENTER (US) 2024-06-25 US disclosed
EP-3104939-B1 TREATMENT OF HEART ATTACK AND ISCHEMIC INJURY WITH SODIUM IODIDE FRED HUTCHINSON CANCER CENTER (US) 2024-05-01 EP disclosed
EP-3347343-B1 AZETIDINIMINES AS CARBAPENEMASES INHIBITORS CENTRE NAT RECH SCIENT (FR) 2023-09-27 EP disclosed
US-11649477-B2 Assays and reagents for antimicrobial susceptibility testing SeLux Diagnostics, Inc. (US) 2023-05-16 US disclosed
CN-109072280-B Method for rapid antimicrobial sensitivity testing 赛录科试诊断公司 2022-10-14 CN disclosed
US-20220313730-A1 HALOGEN TREATMENT OF HEART ATTACK AND ISCHEMIC INJURY FRED HUTCHINSON CANCER CENTER 2022-10-06 US disclosed
US-11339418-B2 Antimicrobial susceptibility testing and microbial identification SeLux Diagnostics, Inc. (US) 2022-05-24 US disclosed
US-11285133-B2 2- or 3-imidazolines as carbapenemases inhibitors CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2022-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12203124-B2 Methods for improved rapid antimicrobial susceptibility testing AMPD3, AMPD1, AMPD2 KDM4E 4444/4885HTT 3276/4885HSP90AA1 127/4885
US-11285133-B2 2- or 3-imidazolines as carbapenemases inhibitors PADI3, PADI1, RPIA KDM4E 1162/4885HTT 4767/4885HSP90AA1 3910/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.