SCHEMBL2953442

SCHEMBL2953442

CCN1CCC(Oc2ccc(-c3nc4c(N)nc(N)nc4[nH]3)c(C)c2)C1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 13/20 0.42
PARP1 P09874 2/20 0.40
ADORA2A P29274 1/20 0.36
ESR1 P03372 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
JAK3 P52333 1/20 0.36
CHEK1 O14757 1/20 0.35
HSP90AB1 P08238 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946524 0.84 HRH4 (0.43) HRH4JAK2JAK1JAK3CHEK1
SCHEMBL2953250 0.81 CARM1 (0.40) HRH4ADORA2ACHEK1
SCHEMBL2953453 0.75 CRHR1 (0.40) PARP1ADORA2AESR1
SCHEMBL2952310 0.74 NPC1 (0.50) HRH4ADORA2A
SCHEMBL2955314 0.74 HRH3 (0.47) PARP1ADORA2AESR1
SCHEMBL2950517 0.73 ADORA2A (0.40) ADORA2ACHEK1
SCHEMBL2955281 0.70 CAMKK2 (0.45) PARP1ADORA2AJAK2JAK1JAK3
SCHEMBL4348402 0.68 HRH3 (0.57) PARP1ESR1
SCHEMBL2951931 0.68 PRKDC (0.42) ADORA2A
SCHEMBL2954446 0.67 TTK (0.37) PARP1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed