SCHEMBL2953250

SCHEMBL2953250

CCN1CCC(c2ccc(-c3nc4c(N)nc(N)nc4[nH]3)c(C)c2)CC1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 6/20 0.40
TLR9 Q9NR96 5/20 0.39
TLR7 Q9NYK1 4/20 0.39
TLR8 Q9NR97 2/20 0.39
CHEK1 O14757 1/20 0.36
FASN P49327 1/20 0.36
HRH4 Q9H3N8 3/20 0.35
DRD2 P14416 1/20 0.34
SLC6A4 P31645 1/20 0.34
DHFR P00374 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946218 0.87 CHEK1 (0.47) CARM1TLR9TLR7TLR8CHEK1
SCHEMBL2946524 0.82 HRH4 (0.43) CHEK1HRH4
SCHEMBL2953442 0.81 HRH4 (0.42) CHEK1HRH4ADORA2A
SCHEMBL2950517 0.79 ADORA2A (0.40) CARM1CHEK1DRD2ADORA2A
SCHEMBL2955281 0.73 CAMKK2 (0.45) TLR7TLR8ADORA2A
SCHEMBL2953257 0.72 CDK1 (0.42) TLR9TLR7TLR8DRD2SLC6A4
SCHEMBL2951931 0.71 PRKDC (0.42) DHFRADORA2AADORA1
SCHEMBL2946339 0.70 CARM1 (0.41) CARM1TLR9TLR7TLR8CHEK1
SCHEMBL2946549 0.69 CDK1 (0.32) HRH4DHFRADORA2AADORA1
SCHEMBL2946541 0.69 CDK1 (0.41) DHFRADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed