SCHEMBL2953453

SCHEMBL2953453

CCN1CCC(Oc2ccc(-n3cnc4c(N)nc(N)nc43)c(C)c2)C1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 1/20 0.40
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
ESR1 P03372 1/20 0.36
PARP1 P09874 1/20 0.35
ACACB O00763 9/20 0.35
ROCK1 Q13464 3/20 0.35
ROCK2 O75116 1/20 0.35
KCNH2 Q12809 1/20 0.35
ADORA2A P29274 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
PI4KA P42356 1/20 0.33
PI4K2B Q8TCG2 1/20 0.33
PI4K2A Q9BTU6 1/20 0.33
PI4KB Q9UBF8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946534 0.84 CRHR1 (0.41) CRHR1CDK1CCNB1CCNE1CDK2
SCHEMBL2953257 0.80 CDK1 (0.42) CRHR1CDK1CCNB1CCNE1CDK2
SCHEMBL2953442 0.75 HRH4 (0.42) ESR1PARP1ADORA2A
SCHEMBL2952316 0.74 NPC1 (0.51) ADORA2A
SCHEMBL2955314 0.73 HRH3 (0.47) ESR1PARP1ACACBADORA2AHRH3
SCHEMBL2946224 0.72 CDK1 (0.40) CDK1CCNB1CCNE1CDK2KCNH2
SCHEMBL2950527 0.72 ADORA2A (0.42) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL2950165 0.70 TLR7 (0.41) CDK1CCNB1CCNE1CDK2PI4KA
SCHEMBL2955288 0.69 TLR7 (0.42) CDK1CCNB1CCNE1CDK2PI4KA
SCHEMBL2951209 0.68 KDM4E (0.42) CDK1CCNB1CCNE1CDK2PI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed