SCHEMBL2953601

SCHEMBL2953601

CCOc1cc(CN2CCOCC2)ccc1-c1nc2c(N)nc(N)nc2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.42
TLR7 Q9NYK1 6/20 0.41
ADORA2A P29274 1/20 0.41
INSR P06213 1/20 0.40
ALK Q9UM73 1/20 0.40
HTT P42858 1/20 0.40
CHEK1 O14757 1/20 0.39
CDK1 P06493 2/20 0.39
CDK2 P24941 2/20 0.39
CDK9 P50750 2/20 0.39
CASP3 P42574 1/20 0.39
CASP7 P55210 1/20 0.39
ILK Q13418 1/20 0.39
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946044 0.86 MAPT (0.43) ADORA2AINSRALKCHEK1CDK1
SCHEMBL2955281 0.85 CAMKK2 (0.45) PARP1TLR7ADORA2AINSRHTT
SCHEMBL2952943 0.76 MAP2K7 (0.45) INSRALKCHEK1
SCHEMBL2953607 0.75 TLR7 (0.44) PARP1TLR7ADORA2AHTTCDK1
SCHEMBL2952310 0.74 NPC1 (0.50) ADORA2AINSRMEN1NPC1RAB9A
SCHEMBL1748552 0.73 SSTR5 (0.48) MEN1KMT2A
SCHEMBL4764968 0.73 HTT (0.52) PARP1HTTMEN1NPC1TP53
SCHEMBL2951931 0.72 PRKDC (0.42) ADORA2AHTTCDK1CDK2MEN1
SCHEMBL2946368 0.68 PRKDC (0.40) ADORA2ACDK1CDK2NPC1TP53
SCHEMBL6557155 0.67 DHFR (0.54) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed