Resminostat

Resminostat

SCHEMBL295540

CN(C)Cc1ccc(S(=O)(=O)n2ccc(/C=C/C(=O)NO)c2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 18/20 1.00
HDAC6 Q9UBN7 15/20 1.00
HDAC3 O15379 8/20 0.98
HDAC8 Q9BY41 6/20 0.98
HDAC2 Q92769 13/20 0.53
HDAC4 P56524 5/20 0.49
MEF2D Q14814 1/20 0.49
HDAC10 Q969S8 5/20 0.45
HDAC11 Q96DB2 4/20 0.45
HDAC9 Q9UKV0 4/20 0.45
KDM1A O60341 1/20 0.45
HDAC5 Q9UQL6 4/20 0.43
HDAC7 Q8WUI4 3/20 0.43
ABL1 P00519 1/20 0.43
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
INSR P06213 1/20 0.43
PDGFRB P09619 1/20 0.43
BRD4 O60885 1/20 0.42
BRD2 P25440 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Resminostat SCHEMBL295541 1.00 HDAC1 (1.00) HDAC1HDAC6HDAC3HDAC8HDAC2
Resminostat SCHEMBL1887878 0.99 HDAC1 (1.00) HDAC1HDAC6HDAC3HDAC8HDAC2
Resminostat SCHEMBL1887874 0.99 HDAC1 (1.00) HDAC1HDAC6HDAC3HDAC8HDAC2
Resminostat SCHEMBL299843 0.98 HDAC1 (0.96) HDAC1HDAC6HDAC3HDAC8HDAC2
Resminostat SCHEMBL299845 0.98 HDAC1 (0.96) HDAC1HDAC6HDAC3HDAC8HDAC2
Resminostat SCHEMBL299686 0.97 HDAC1 (0.94) HDAC1HDAC6HDAC3HDAC8HDAC2
Resminostat SCHEMBL299688 0.97 HDAC1 (0.94) HDAC1HDAC6HDAC3HDAC8HDAC2
SCHEMBL3149324 0.97 HDAC1 (0.94) HDAC1HDAC6HDAC3HDAC8HDAC2
SCHEMBL3149313 0.97 HDAC1 (0.94) HDAC1HDAC6HDAC3HDAC8HDAC2
Resminostat SCHEMBL299597 0.96 HDAC1 (0.92) HDAC1HDAC6HDAC3HDAC8HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1778 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026107052-A1 COMBINATION TREATMENTS USING EPIGENETIC INHIBITION AND SYNGRI-MEDIATED FRATAXIN EXPRESSION ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2026-05-21 WO claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
EP-4720316-A2 NON-VIRAL CELL ENGINEERING Arsenal Biosciences, Inc. (US) 2026-04-08 EP claimed
US-12582635-B2 Compositions and methods for treating cancer with atypical BRAF mutations BIOMED VALLEY DISCOVERIES, INC. (US) 2026-03-24 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
US-20250381202-A1 PRODRUG KIT FOR MULTI-PRONGED CHEMOTHERAPY ZOUNEK ALEX (DE) 2025-12-18 US claimed
WO-2025235998-A1 PLURIPOTENT STEM CELL DERIVED MESENCHYMAL STEM CELLS WITH ENHANCED IMMUNE MODULATORY ACTIVITY IMMORTA BIO, INC. (US) 2025-11-13 WO claimed
US-20250339551-A1 AN ANTIBODY-DRUG CONJUGATE HAVING TWO OR MORE DIFFERENT FUNCTIONAL SMALL MOLECULES FOR ENHANCED TREATMENT OF REFRACTORY DISEASES HANGZHOU SEEHE BIOTECHNOLOGY CO., LTD (CN) 2025-11-06 US claimed
EP-4642484-A1 TARGETED TREATMENT OF PROSTATE CANCERS AND OTHER TUMORS BY AN ANTIBODY-DRUG CONJUGATE Hangzhou Seehe Biotechnology Co., Ltd (CN) 2025-11-05 EP claimed
CN-101287706-A Sulphonylpyrrole hydrochloride salts as histone deacetylases inhibitors NYCOMED GMBH (DE) 2008-10-15 CN claimed
CN-101268070-A Novel sulphonylpyrroles as inhibitors of HDAC novel sulphonylpyrroles NYCOMED GMBH (DE) 2008-09-17 CN claimed
EP-1928872-A1 NOVEL SULPHONYLPYRROLES AS INHIBITORS OF HDAC S NOVEL SULPHONYLPYRROLES Nycomed GmbH (DE) 2008-06-11 EP claimed
EP-1928826-A1 SULPHONYLPYRROLE HYDROCHLORIDE SALTS AS HISTONE DEACETYLASES INHIBITORS Nycomed GmbH (DE) 2008-06-11 EP claimed
US-20070184979-A1 Novel sulfonylpyrroles ALTANA PHARMA AG (DE) 2007-08-09 US claimed
WO-2007039404-A1 NOVEL SULPHONYLPYRROLES AS INHIBITORS OF HDAC S NOVEL SULPHONYLPYRROLES NYCOMED GMBH (DE) 2007-04-12 WO claimed
WO-2007039403-A1 SULPHONYLPYRROLE HYDROCHLORIDE SALTS AS HISTONE DEACETYLASES INHIBITORS NYCOMED GMBH (DE) 2007-04-12 WO claimed
CN-1926103-A Sulfonyl pyrroles as HDAC inhibitors ALTANA PHARMA AG (DE) 2007-03-07 CN claimed
EP-1725528-A2 SULPHONYLPYRROLES AS HDAC INHIBITORS Altana Pharma AG (DE) 2006-11-29 EP claimed
WO-2005087724-A2 SULPHONYLPYRROLES AS HDAC INHIBITORS ALTANA PHARMA AG (DE) 2005-09-22 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250381202-A1 PRODRUG KIT FOR MULTI-PRONGED CHEMOTHERAPY KIT, CTSL, PAICS HDAC1 517/4885HDAC6 1590/4885HDAC3 1207/4885
US-20250339551-A1 AN ANTIBODY-DRUG CONJUGATE HAVING TWO OR MORE DIFFERENT FUNCTIONAL SMALL MOLECULES FOR ENHANCED TREATMENT OF REFRACTORY DISEASES FCGR2A, FCGR3B, FCGR1A HDAC1 2078/4885HDAC6 102/4885HDAC3 1362/4885
US-20070184979-A1 Novel sulfonylpyrroles HDAC1, HDAC4, HDAC3 HDAC1 1/4885HDAC6 8/4885HDAC3 3/4885
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule CD4, TAP1, MCTS1 HDAC1 2312/4885HDAC6 814/4885HDAC3 3198/4885
US-12582635-B2 Compositions and methods for treating cancer with atypical BRAF mutations BRAF, SRMS, MAPK3 HDAC1 3880/4885HDAC6 4490/4885HDAC3 2618/4885
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES WNT3A, GSK3B, GSK3A HDAC1 71/4885HDAC6 665/4885HDAC3 97/4885
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS DCLRE1A, CCR3, CCR8 HDAC1 1894/4885HDAC6 920/4885HDAC3 708/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.