Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | KDM4E | B2RXH2 | 8/20 | 0.42 |
| ▸ | MEN1 | O00255 | 2/20 | 0.42 |
| ▸ | KMT2A | Q03164 | 2/20 | 0.42 |
| ▸ | ALDH1A1 | P00352 | 6/20 | 0.39 |
| ▸ | LMNA | P02545 | 3/20 | 0.39 |
| ▸ | CYP3A4 | P08684 | 1/20 | 0.39 |
| ▸ | MAPT | P10636 | 1/20 | 0.39 |
| ▸ | TSHR | P16473 | 1/20 | 0.39 |
| ▸ | BLM | P54132 | 1/20 | 0.39 |
| ▸ | PMP22 | Q01453 | 1/20 | 0.39 |
| ▸ | HPGD | P15428 | 6/20 | 0.38 |
| ▸ | HSD17B10 | Q99714 | 2/20 | 0.38 |
| ▸ | CYP2C9 | P11712 | 1/20 | 0.38 |
| ▸ | APAF1 | O14727 | 1/20 | 0.38 |
| ▸ | CASP6 | P55212 | 1/20 | 0.38 |
| ▸ | GAA | P10253 | 2/20 | 0.36 |
| ▸ | PKM | P14618 | 1/20 | 0.36 |
| ▸ | GLA | P06280 | 1/20 | 0.35 |
| ▸ | SMN1; SMN2 | Q16637 | 1/20 | 0.34 |
| ▸ | CNOT7 | Q9UIV1 | 1/20 | 0.34 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL169145 | 0.87 | KDM4E (0.41) | KDM4EMEN1KMT2AALDH1A1LMNA | |
| SCHEMBL7367989 | 0.81 | ALDH1A1 (0.46) | KDM4EMEN1KMT2AALDH1A1LMNA | |
| SCHEMBL2948723 | 0.79 | GAA (0.53) | KDM4EMEN1KMT2AALDH1A1TSHR | |
| SCHEMBL3489068 | 0.78 | PNP (0.44) | MEN1KMT2AALDH1A1LMNACYP3A4 | |
| SCHEMBL7419700 | 0.76 | ALDH1A1 (0.46) | KDM4EKMT2AALDH1A1GAA | |
| SCHEMBL9199287 | 0.75 | LMNA (0.40) | KDM4EMEN1KMT2AALDH1A1LMNA | |
| SCHEMBL515776 | 0.73 | ALDH1A1 (0.54) | KDM4EMEN1KMT2AALDH1A1LMNA | |
| SCHEMBL10432471 | 0.72 | HSD17B10 (0.49) | KDM4EMEN1KMT2AALDH1A1LMNA | |
| SCHEMBL16359618 | 0.68 | ADORA2A (0.45) | MEN1KMT2AALDH1A1SMN1; SMN2 | |
| SCHEMBL9299928 | 0.68 | LMNA (0.60) | ALDH1A1LMNACYP3A4MAPTTSHR |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-8957020-B2 | Mnk kinase homologous proteins involved in the regulation of energy homeostasis and organelle metabolism | BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) | 2015-02-17 | — | — | US | disclosed |
| US-8828934-B2 | Mnk kinase homologous proteins involved in the regulation of energy homeostasis and organelle metabolism | BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) | 2014-09-09 | — | — | US | disclosed |
| US-20140213510-A1 | USE OF PLEITROPHIN FOR PREVENTING AND TREATING PANCREATIC DISEASES AND/OR OBESITY AND/OR METABOLIC SYNDROME | EVOTEC INTERNATIONAL GMBH (DE) | 2014-07-31 | — | — | US | disclosed |
| EP-2289908-B1 | Use of DG177 secreted protein products for preventing and treating pancreatic diseases and/or obesity and/or metabolic syndrome | EVOTEC INTERNAT GMBH (DE) | 2013-08-07 | — | — | EP | disclosed |
| US-8501473-B2 | Use of pleitrophin for preventing and treating pancreatic diseases and/or obesity and/or metabolic syndrome | EVOTEC INTERNATIONAL GMBH (DE) | 2013-08-06 | — | — | US | disclosed |
| EP-1605965-B1 | USE OF SAPOSIN-RELATED PROTEINS FOR PREVENTING AND TREATING OBESITY, DIABETES AND/OR METABOLIC SYNDROME | DEVELOGEN AG (DE) | 2012-12-26 | — | — | EP | disclosed |
| EP-1644406-B1 | USE OF DG153 SECRETED PROTEIN PRODUCTS FOR PREVENTING AND TREATING PANCREATIC DISEASES AND/OR OBESITY AND/OR METABOLIC SYNDROME | DEVELOGEN AG (DE) | 2012-08-15 | — | — | EP | disclosed |
| EP-2096120-B1 | Use of secreted protein products for preventing and treating pancreatic diseases and/or obesity and/or metabolic syndrome | DEVELOGEN AG (DE) | 2012-03-14 | — | — | EP | disclosed |
| US-20120045452-A1 | Mnk KINASE HOMOLOGOUS PROTEINS INVOLVED IN THE REGULATION OF ENERGY HOMEOSTASIS AND ORGANELLE METABOLISM | DEVELOGEN AKTIENGESELLSCHAFT FUER ENTWICKLUNGSBIOLOGISCHE FORSCHUNG (DE) | 2012-02-23 | — | — | US | disclosed |
| US-20120045451-A1 | Mnk KINASE HOMOLOGOUS PROTEINS INVOLVED IN THE REGULATION OF ENERGY HOMEOSTASIS AND ORGANELLE METABOLISM | DEVELOGEN AKTIENGESELLSCHAFT FUER ENTWICKLUNGSBIOLOGISCHE FORSCHUNG (DE) | 2012-02-23 | — | — | US | disclosed |
| WO-2004031392-A1 | MIPP1 HOMOLOGOUS NUCLEIC ACIDS AND PROTEINS INVOLVED IN THE REGULATION OF ENERGY HOMEOSTATIS | DeveloGen Aktiengesellschaft für entwicklungsbiologische Forschung (DE) | 2004-04-15 | — | — | WO | disclosed |
| WO-2004028554-A2 | SKRP, ASTRAY, STRING, VACM ASSOCIATED WITH METABOLIC CONTROL | DeveloGen Aktiengesellschaft für entwicklungsbiologische Forschung (DE) | 2004-04-08 | — | — | WO | disclosed |
| WO-2004022089-A1 | MINIBRAIN HOMOLOGOUS PROTEINS INVOLVED IN THE REGULATION OF ENERGY HOMEOSTASIS | DeveloGen Aktiengesellschaft für entwicklungsbiologische Forschung (DE) | 2004-03-18 | — | — | WO | disclosed |
| WO-2004020465-A2 | PROTEINS INVOLVED IN THE REGULATION OF ENERGY HOMEOSTASIS | DeveloGen Aktiengesellschaft für entwicklungsbiologische Forschung (DE) | 2004-03-11 | — | — | WO | disclosed |
| WO-2004016641-A2 | PROTEINS INVOLVED IN THE REGULATION OF ENERGY HOMEOSTASIS | DeveloGen Aktiengesellschaft für entwicklungsbiologische Forschung (DE) | 2004-02-26 | — | — | WO | disclosed |
| WO-2004012758-A1 | USE OF TGF BETA IG-H3 FOR PREVENTING AND TREATING OBESITY, DIABETES AND/OR METABOLIC SYNDROME | DeveloGen Aktiengesellschaft für entwicklungsbiologische Forschung (DE) | 2004-02-12 | — | — | WO | disclosed |
| WO-2003074078-A2 | CG3842 HOMOLOGOUS PROTEINS INVOLVED IN THE REGULATION OF ENERGY HOMEOSTASIS | DeveloGen Aktiengesellschaft für entwicklungsbiologische Forschung (DE) | 2003-09-12 | — | — | WO | disclosed |
| WO-2003047611-A2 | PTP10D, TEC AND EDTP INVOLVED IN TRIGLYCERID-METABOLISM | DeveloGen Aktiengesellschaft für entwicklungsbiologische Forschung (DE) | 2003-06-12 | — | — | WO | disclosed |
| WO-2003039574-A1 | ENDOPHILIN HOMOLOGOUS PROTEINS INVOLVED IN THE REGULATION OF ENERGY HOMEOSTASIS | DEVELOGEN AKTIENGESELLSCHAFT FÜR ENTIWICKLUNGSBIOLOGISCHE FORSCHUNG (DE) | 2003-05-15 | — | — | WO | disclosed |
| WO-2003037362-A2 | MNK KINASE HOMOLOGOUS PROTEINS INVOLVED IN THE REGULATION OF ENERGY HOMEOSTASIS AND ORGANELLE METABOLISM | DeveloGen Aktiengesellschaft für entwicklungsbiologische Forschung (DE) | 2003-05-08 | — | — | WO | disclosed |