SCHEMBL29620451

SCHEMBL29620451

O=C1c2ccncc2CN1CCF

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
USP19 O94966 1/20 0.39
NPSR1 Q6W5P4 1/20 0.37
CYP11B2 P19099 1/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
ACHE P22303 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
HTR1A P08908 2/20 0.35
DRD2 P14416 2/20 0.35
DRD5 P21918 1/20 0.35
DRD3 P35462 1/20 0.35
HTR7 P34969 1/20 0.34
DHPS P49366 1/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15164719 0.84 PKN2 (0.42) KDM4EALOX15TSHRSIRT1USP19
SCHEMBL29620463 0.84 KDM4E (0.43) KDM4EALOX15TSHRSIRT1USP19
SCHEMBL29620459 0.81 IDH1 (0.40) KDM4EALOX15TSHRSIRT1USP19
SCHEMBL29620469 0.81 ALDH1A1 (0.49) KDM4EALOX15TSHRSIRT1NPSR1
SCHEMBL29620441 0.80 USP19 (0.42) KDM4EALOX15TSHRSIRT1USP19
SCHEMBL29620429 0.80 USP19 (0.39) KDM4EALOX15TSHRSIRT1USP19
SCHEMBL30947594 0.75 CYP11B2 (0.41) KDM4ETSHRUSP19NPSR1CYP11B2
SCHEMBL11923831 0.75 CYP11B2 (0.41) NPSR1CYP11B2PDE3BPDE3A
SCHEMBL29620473 0.74 ALOX15 (0.36) KDM4EALOX15TSHRUSP19NPSR1
SCHEMBL31667471 0.74 DHPS (0.46) DHPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4041732-A1 ISO-CITRATE DEHYDROGENASE (IDH) INHIBITOR ZHEJIANG METON PHARMACEUTICAL CO., LTD (CN) 2022-08-17 EP claimed
CN-114555597-A Isocitrate Dehydrogenase (IDH) inhibitors 浙江迈同生物医药有限公司 2022-05-27 CN claimed