SCHEMBL29623436

SCHEMBL29623436

Fc1ccc(Oc2cccc(Br)c2)cc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 7/20 0.47
CDK8 P49336 1/20 0.43
HTR2A P28223 1/20 0.42
SLC6A4 P31645 1/20 0.42
KCNH2 Q12809 1/20 0.42
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ATM Q13315 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAOB P27338 3/20 0.40
TLR8 Q9NR97 1/20 0.38
SCN9A Q15858 1/20 0.36
EGFR P00533 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14649871 0.83 AR (0.49) ARCDK8CYP1A2CYP3A4CYP2D6
SCHEMBL3839157 0.76 ALDH1A1 (0.54) MAOBEGFR
SCHEMBL3838974 0.76 ALDH1A1 (0.54) MAOBEGFR
SCHEMBL457828 0.76 MAOB (0.54) SLC6A4MAOBEGFR
SCHEMBL29623526 0.76 CYP1A2 (0.45) ARCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9546439 0.76 NPSR1 (0.53) SLC6A4CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL29603301 0.76 NPSR1 (0.53) SLC6A4CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL2394719 0.75 MAOB (0.59) CDK8CYP1A2CYP2C9CYP2C19MAOB
SCHEMBL29623441 0.75 NPSR1 (0.56) HTR2ASLC6A4KCNH2CYP1A2CYP3A4
SCHEMBL31360383 0.75 CETP (0.43) SLC6A4CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109790149-B Phenoxytriazoles 豪夫迈·罗氏有限公司 2022-05-17 CN disclosed