SCHEMBL29645914

SCHEMBL29645914

O=c1nccccc1Nc1nc2c(C(F)(F)F)cccc2c2nc(-c3ccc(Cl)cc3)nn12

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 6/20 0.40
NR1H3 Q13133 6/20 0.40
ADORA3 P0DMS8 7/20 0.40
ADORA2A P29274 4/20 0.39
ADORA1 P30542 3/20 0.39
MAPT P10636 1/20 0.38
P2RX7 Q99572 1/20 0.35
USP1 O94782 1/20 0.35
WDR48 Q8TAF3 1/20 0.35
XDH P47989 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645682 0.92 ADORA3 (0.40) NR1H2NR1H3ADORA3ADORA2AADORA1
SCHEMBL31149976 0.91 ADORA3 (0.38) NR1H2NR1H3ADORA3ADORA2AADORA1
SCHEMBL29645803 0.90 POLB (0.46) ADORA3ADORA2AADORA1MAPTP2RX7
SCHEMBL29646148 0.87 LMNA (0.39) MAPT
SCHEMBL29645755 0.86 MAPT (0.40) ADORA3ADORA2AADORA1MAPTXDH
SCHEMBL29645837 0.85 EGFR (0.36) P2RX7XDH
SCHEMBL29645723 0.85 P2RX7 (0.36) P2RX7
SCHEMBL29645738 0.84 NTRK1 (0.36) ADORA3ADORA2AADORA1P2RX7
SCHEMBL29645600 0.84 PDK2 (0.32) ADORA3ADORA2AADORA1P2RX7
SCHEMBL29645888 0.83 MAPT (0.55) ADORA3ADORA2AADORA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed