SCHEMBL29645837

SCHEMBL29645837

O=c1nccccc1Nc1nc2c(C(F)(F)F)cccc2c2nc(-c3cn[nH]c3)nn12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.36
SLC40A1 Q9NP59 1/20 0.34
PSEN1 P49768 2/20 0.33
PSEN2 P49810 2/20 0.33
APH1B Q8WW43 2/20 0.33
NCSTN Q92542 2/20 0.33
APH1A Q96BI3 2/20 0.33
PSENEN Q9NZ42 2/20 0.33
P2RX7 Q99572 4/20 0.33
JAK2 O60674 1/20 0.32
CDK1 P06493 2/20 0.32
DYRK3 O43781 1/20 0.32
PRKD3 O94806 1/20 0.32
MAP4K4 O95819 1/20 0.32
CDK2 P24941 1/20 0.32
FLT4 P35916 1/20 0.32
CSNK1D P48730 1/20 0.32
CLK2 P49760 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645807 0.87 TP53 (0.39) SLC40A1P2RX7CDK2ROCK2ROCK1
SCHEMBL29645682 0.86 ADORA3 (0.40) P2RX7XDHTP53SMN1; SMN2RXFP1
SCHEMBL29645803 0.85 POLB (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL29645914 0.85 NR1H2 (0.40) P2RX7XDH
SCHEMBL29645600 0.85 PDK2 (0.32) SLC40A1PSEN1PSEN2APH1BNCSTN
SCHEMBL29646148 0.84 LMNA (0.39) CSNK1DTP53RXFP1
SCHEMBL29645878 0.84 HSP90AA1 (0.35) SLC40A1PSEN1PSEN2APH1BNCSTN
SCHEMBL29645654 0.84 MAPT (0.43) POLBTP53SMN1; SMN2RXFP1
SCHEMBL29645745 0.84 PSEN1 (0.34) SLC40A1PSEN1PSEN2APH1BNCSTN
SCHEMBL29645738 0.82 NTRK1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed