SCHEMBL29699666

SCHEMBL29699666

CON(C)C(=O)c1cccc(C(F)(F)F)c1C

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 1/20 0.46
CTSS P25774 2/20 0.44
MLYCD O95822 1/20 0.42
DHODH Q02127 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MAOB P27338 1/20 0.40
GPBAR1 Q8TDU6 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
EPHX2 P34913 1/20 0.38
KCNK3 O14649 2/20 0.38
KCNK9 Q9NPC2 2/20 0.38
MAPT P10636 2/20 0.38
HDAC8 Q9BY41 1/20 0.38
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15761208 1.00 TAS2R14 (0.46) TAS2R14CTSSMLYCDDHODHHDAC6
SCHEMBL1125455 0.86 HDAC8 (0.49) TAS2R14CTSSMLYCDMAOBGPBAR1
SCHEMBL8575500 0.86 LMNA (0.49) MLYCDMAOBGPBAR1SMN1; SMN2LMNA
SCHEMBL21401288 0.80 ESR1 (0.55) MLYCDSMN1; SMN2GAAALDH1A1
SCHEMBL30577974 0.79 MLYCD (0.42) CTSSMLYCDMAOBGPBAR1SMN1; SMN2
SCHEMBL726068 0.78 TAS2R14 (0.54) TAS2R14CTSSDHODHHDAC6LMNA
SCHEMBL16625279 0.77 CTSS (0.51) TAS2R14CTSSMLYCDDHODHHDAC6
SCHEMBL28052031 0.77 TAS2R14 (0.55) TAS2R14CTSSDHODHHDAC6LMNA
SCHEMBL4837622 0.76 KMT2A (0.41) MLYCDSMN1; SMN2LMNAALDH1A1
SCHEMBL14381951 0.76 ESR1 (0.36) MLYCDMAOBSMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116655625-A Compounds as SOS1 inhibitors and uses thereof 南京圣和药业股份有限公司 2023-08-29 CN disclosed
CN-115785088-A Compounds as SOS1 inhibitors and uses thereof 南京圣和药业股份有限公司 2023-03-14 CN disclosed
CN-114685488-A Compounds as SOS1 inhibitors and uses thereof 南京圣和药业股份有限公司 2022-07-01 CN disclosed