SCHEMBL2970574

SCHEMBL2970574

Cc1cc(Br)c(N)c([N+](=O)[O-])c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.63
CYP3A4 P08684 5/20 0.63
GPR35 Q9HC97 1/20 0.53
TSHR P16473 4/20 0.53
CTSB P07858 1/20 0.51
CYP1A2 P05177 2/20 0.44
RECQL P46063 1/20 0.44
KDM4E B2RXH2 2/20 0.43
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
MAPT P10636 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 1/20 0.41
G6PD P11413 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2232801 0.87 GPR35 (0.61) ALDH1A1CYP3A4GPR35TSHRCTSB
SCHEMBL27561588 0.82 GPR35 (0.55) ALDH1A1CYP3A4GPR35TSHRCYP1A2
SCHEMBL22968279 0.82 GPR35 (0.55) ALDH1A1CYP3A4GPR35TSHRCYP1A2
SCHEMBL7786697 0.82 TSHR (0.60) ALDH1A1CYP3A4GPR35TSHRCYP1A2
SCHEMBL349045 0.82 GPR35 (0.55) ALDH1A1CYP3A4GPR35TSHRCYP1A2
SCHEMBL29816776 0.82 GPR35 (0.55) ALDH1A1CYP3A4GPR35TSHRCYP1A2
SCHEMBL2783704 0.79 ALDH1A1 (0.68) ALDH1A1CYP3A4TSHRCTSBKDM4E
SCHEMBL29706644 0.79 ALDH1A1 (0.68) ALDH1A1CYP3A4TSHRCTSBKDM4E
SCHEMBL11539985 0.79 GPR35 (0.68) ALDH1A1CYP3A4GPR35TSHRCYP1A2
SCHEMBL22232253 0.78 GPR35 (0.52) ALDH1A1CYP3A4GPR35TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 99 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025171194-A9 CRYSTALLINE FORMS OF (R)-6-CHLORO-3-((1-(2-CYANO-7-METHYL-3-MORPHOLINOQUINOXALIN-5-YL)ETHYL)AMINO)PICOLINIC ACID Mirati Therapeutics, Inc. (US) 2026-05-21 WO disclosed
EP-4709714-A1 SUBSTITUTED QUINOXALINES Mirati Therapeutics, Inc. (US) 2026-03-18 EP disclosed
CN-121586713-A Quinoline derivatives and pharmaceutical compositions thereof for the treatment of diseases 百济神州(苏州)生物科技有限公司 2026-02-27 CN disclosed
US-12545639-B2 3-substituted phenylamidine compounds, preparation and use thereof PI INDUSTRIES LTD. (IN) 2026-02-10 US disclosed
US-12528827-B2 Tricyclic heteroaryl-substituted quinoline and azaquinoline compounds as PAR4 inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2026-01-20 US disclosed
EP-4647426-A2 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS, PREPARATION AND USE THEREOF PI Industries Ltd. (IN) 2025-11-12 EP disclosed
US-20250276960-A1 CRYSTALLINE FORMS OF (R)-6-CHLORO-3-((1-(2-CYANO-7-METHYL-3-MORPHOLINOQUINOXALIN-5-YL)ETHYL)AMINO)PICOLINIC ACID Mirati Therapeutics, Inc. (US) 2025-09-04 US disclosed
EP-4596551-A1 COMPOUNDS WITH ANTI-KRAS MUTANT TUMOR ACTIVITY Trasveda Ltd. (KY) 2025-08-06 EP disclosed
US-20250121073-A1 IRAK DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2025-04-17 US disclosed
WO-2025021217-A1 QUINOLINE DERIVATIVES AND PHARMARCEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF DISEASE BEIGENE SWITZERLAND GMBH (CH) 2025-01-30 WO disclosed
EP-0559843-B1 SUBSTITUTED N-HETEROBICYCLIC HERBICIDES DU PONT (US) 1994-09-14 EP disclosed
EP-0559843-A1 SUBSTITUTED N-HETEROBICYCLIC HERBICIDES. DU PONT (US) 1993-09-15 EP disclosed
WO-1992009578-A1 SUBSTITUTED FUSED HETEROCYCLIC HERBICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-06-11 WO disclosed
US-5110347-A Pre- and postemergence; quinoxaline derivatives E. I DU PONT DE NEMOURS AND COMPANY (US) 1992-05-05 US disclosed
US-4479899-A OF POLYESTERS BAYER AKTIENGESELLSCHAFT (DE) 1984-10-30 US disclosed
US-4452609-A Dyeing red with 2,6-dicyano-2'-sulfonamido-4'-amino-azo-benzenes BAYER AKTIENGESELLSCHAFT (DE) 1984-06-05 US disclosed
US-4237048-A COLORFASTNESS; FOR DYEING NATURAL AND SYNTHETIC FIBERS BAYER AKTIENGESELLSCHAFT (DE) 1980-12-02 US disclosed
US-4105655-A PHENYL-AZO-ANILINO DYESTUFF BAYER AKTIENGESELLSCHAFT (DE) 1978-08-08 US disclosed
US-4083844-A Phenylazo orthocyano phenylazo or orthocyano phenylazo phenylazo containing dyestuffs BAYER AKTIENGESELLSCHAFT (DT) 1978-04-11 US disclosed
US-3962209-A PROCESS FOR PREPARING AZO DYESTUFFS WITH ORTHO-AZO CYANO GROUPS BY CYANO EXCHANGE OF METAL CYANIDES AND HALO DYESTUFFS BAYER AKTIENGESELLSCHAFT (DT) 1976-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250276960-A1 CRYSTALLINE FORMS OF (R)-6-CHLORO-3-((1-(2-CYANO-7-METHYL-3-MORPHOLINOQUINOXALIN-5-YL)ETHYL)AMINO)PICOLINIC ACID UACA, CA6, CALU ALDH1A1 3833/4885CYP3A4 2869/4885GPR35 3858/4885
US-20250121073-A1 IRAK DEGRADERS AND USES THEREOF IRAK2, IRAK3, IRAK1 ALDH1A1 2776/4885CYP3A4 2542/4885GPR35 3025/4885
US-12545639-B2 3-substituted phenylamidine compounds, preparation and use thereof CBR1, CBR3, HCCS ALDH1A1 2035/4885CYP3A4 264/4885GPR35 3991/4885
US-12528827-B2 Tricyclic heteroaryl-substituted quinoline and azaquinoline compounds as PAR4 inhibitors F2RL3, F2R, PF4 ALDH1A1 1173/4885CYP3A4 23/4885GPR35 2279/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.