SCHEMBL29720591

SCHEMBL29720591

Oc1ccc2scnc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
HSD17B10 Q99714 1/20 0.50
KDM4E B2RXH2 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
HSD11B1 P28845 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HKDC1 Q2TB90 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAP3K11 Q16584 1/20 0.40
NAMPT P43490 1/20 0.40
CA2 P00918 1/20 0.40
MEN1 O00255 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
KMT2A Q03164 1/20 0.39
PTK6 Q13882 2/20 0.39
HPGD P15428 1/20 0.39
ENPP2 Q13822 1/20 0.39
GAA P10253 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL927314 1.00 ALDH1A1 (0.50) ALDH1A1HSD17B10KDM4EL3MBTL1HSD11B1
Hydrochloric Acid SCHEMBL31731478 0.98 ALDH1A1 (0.48) ALDH1A1HSD17B10KDM4EL3MBTL1HSD11B1
SCHEMBL1852870 0.84 FFAR1 (0.48) ALDH1A1HSD17B10MAP3K11MEN1KMT2A
SCHEMBL23069 0.83 NPC1 (0.56) ALDH1A1HSD17B10KDM4EL3MBTL1NPC1
Hydrochloric Acid SCHEMBL27543158 0.81 NPC1 (0.55) ALDH1A1HSD17B10KDM4EL3MBTL1NPC1
SCHEMBL29265410 0.80 ALDH1A1 (0.45) ALDH1A1HSD17B10L3MBTL1HSD11B1NPC1
SCHEMBL13394608 0.80 APP (0.40) ALDH1A1HSD17B10KDM4EL3MBTL1HSD11B1
SCHEMBL30954741 0.80 ALDH1A1 (0.45) ALDH1A1HSD17B10L3MBTL1HSD11B1NPC1
Ethane SCHEMBL27382338 0.79 NPC1 (0.53) ALDH1A1HSD17B10KDM4EL3MBTL1NPC1
SCHEMBL3310695 0.79 L3MBTL1 (0.42) ALDH1A1HSD17B10KDM4EL3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250109139-A1 TRICYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF CENTER FOR EXCELLENCE IN MOLECULAR CELL SCIENCE, CHINESE ACADEMY OF SCIENCES (CN) 2025-04-03 US disclosed
US-20240124456-A1 AZA-ERGOLINE DERIVATIVE AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF SHANGHAITECH UNIVERSITY (CN) 2024-04-18 US disclosed
EP-4286384-A1 AZA-ERGOLINE DERIVATIVE AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF ShanghaiTech University (CN) 2023-12-06 EP disclosed
WO-2022161493-A1 AZA-ERGOLINE DERIVATIVE AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海科技大学 2022-08-04 WO disclosed
CN-114835709-A Aza-ergoline derivative and preparation method and application thereof 上海科技大学 2022-08-02 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240124456-A1 AZA-ERGOLINE DERIVATIVE AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF ERG, CHRNA7, CHRNA5 ALDH1A1 399/4885HSD17B10 1448/4885KDM4E 2460/4885
US-20250109139-A1 TRICYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF PARK7, HADH, BDNF ALDH1A1 1460/4885HSD17B10 677/4885KDM4E 4265/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.