SCHEMBL29777975

SCHEMBL29777975

CN(C)C(=O)c1cccc(OCCN(C)C(=O)OCc2ccccc2)c1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.55
MAOB P27338 1/20 0.50
NR4A2 P43354 1/20 0.49
RAB9A P51151 1/20 0.48
MEN1 O00255 1/20 0.47
ESR1 P03372 4/20 0.46
LTB4R Q15722 1/20 0.46
LTB4R2 Q9NPC1 1/20 0.46
SMPD1 P17405 1/20 0.45
SRD5A2 P31213 1/20 0.44
F10 P00742 1/20 0.44
BRD4 O60885 1/20 0.44
PTPN1 P18031 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24627426 1.00 KMT2A (0.55) KMT2AMAOBNR4A2RAB9AMEN1
SCHEMBL24627541 0.87 EGFR (0.49) KMT2AMAOBNR4A2RAB9AMEN1
SCHEMBL29777992 0.81 L3MBTL1 (0.60) KMT2AMAOBNR4A2RAB9ASMPD1
SCHEMBL29777971 0.78 ALDH1A1 (0.43)
SCHEMBL7367495 0.75 ALDH1A1 (0.58) KMT2A
SCHEMBL9536302 0.75 LTA4H (0.47) LTB4RLTB4R2
SCHEMBL5968220 0.74 RAB9A (0.64) KMT2ARAB9AMEN1ESR1F10
SCHEMBL10466517 0.74 MAOB (0.69) KMT2AMAOBNR4A2MEN1SMPD1
SCHEMBL24627626 0.73 KMT2A (0.51) KMT2AESR1SMPD1F10
SCHEMBL12134478 0.73 ESR1 (0.69) KMT2ARAB9AMEN1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022148879-A1 QUINAZOLINE DERIVATIVES USEFUL AS MODULATORS OF ACKR3 STICHTING VU (NL) 2022-07-14 WO disclosed