SCHEMBL2982804

SCHEMBL2982804

COC(=O)CCCC(=O)NC1CCC(Cc2ccc(F)cc2)(N(C)C)CC1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.39
ACKR3 P25106 1/20 0.39
HRH3 Q9Y5N1 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
CA12 O43570 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2976452 0.90 MEN1 (0.46) CYP1A2CYP3A4CYP2D6CYP2C9HPGD
SCHEMBL2989386 0.89 LMNA (0.45) CYP1A2CYP3A4CYP2D6CYP2C9HPGD
SCHEMBL2985381 0.89 OPRM1 (0.48) CYP1A2CYP3A4CYP2D6CYP2C9HPGD
SCHEMBL2983741 0.88 SIGMAR1 (0.41) ALDH1A1ACKR3OPRM1OPRL1
SCHEMBL2987816 0.84 MEN1 (0.47) LMNAOPRM1OPRL1
SCHEMBL2989227 0.83 BCHE (0.41) HPGDALDH1A1OPRM1OPRL1
SCHEMBL2987319 0.82 MEN1 (0.47) OPRM1OPRL1
SCHEMBL206079 0.82 OPRM1 (0.54) OPRM1OPRL1
SCHEMBL2977995 0.82 THRB (0.48) HPGDOPRM1OPRL1
SCHEMBL4048579 0.80 KMT2A (0.47) ALDH1A1ACKR3OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7786328-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2010-08-31 US claimed
US-20070281954-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-12-06 US claimed
US-7786328-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2010-08-31 US disclosed
US-20070281954-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-12-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070281954-A1 Cyclohexyl-1,4-diamine compounds DPYD, PKD1, AOC1 CYP1A2 100/4885CYP3A4 124/4885CYP2D6 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.