SCHEMBL29860127

SCHEMBL29860127

CCN1CCc2ccc(N)cc2CC1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATAD2 Q6PL18 2/20 0.49
NR1H2 P55055 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
HSD17B10 Q99714 1/20 0.37
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 3/20 0.36
HTR1A P08908 2/20 0.36
HTR7 P34969 1/20 0.36
GFER P55789 1/20 0.36
HPGD P15428 2/20 0.36
HCN4 Q9Y3Q4 1/20 0.35
DRD2 P14416 2/20 0.35
DRD1 P21728 1/20 0.35
HTR2A P28223 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29119500 1.00 ATAD2 (0.49) ATAD2NR1H2MAPK1KMT2AGAA
SCHEMBL2061379 0.81 SMN1; SMN2 (0.57) ATAD2NR1H2MAPK1KMT2AGAA
SCHEMBL1950172 0.80 CASP1 (0.49) ATAD2CASP1CASP7HSD17B10
SCHEMBL885867 0.79 DRD1 (0.54) GAASMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL29119426 0.79 DRD2 (0.50) KMT2AKDM4EALDH1A1MAPTHTR1A
SCHEMBL29119474 0.77 PNMT (0.43) MAPK1KMT2AGAAALDH1A1MAPT
SCHEMBL2267570 0.76 HTR2A (0.45) ATAD2KMT2AGAAKDM4EALDH1A1
SCHEMBL618018 0.76 ATAD2 (0.55) ATAD2KMT2AGAASMN1; SMN2CASP1
SCHEMBL30168583 0.76 ATAD2 (0.55) ATAD2KMT2AGAASMN1; SMN2CASP1
SCHEMBL29119447 0.75 HSP90AA1 (0.48) KMT2AGAAKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116888127-A Tri-fused ring HPK1 inhibitor and application thereof 轩竹生物科技股份有限公司 2023-10-13 CN disclosed
WO-2022188823-A1 TRICYCLIC HPK1 INHIBITOR AND USE THEREOF 山东轩竹医药科技有限公司 2022-09-15 WO disclosed