SCHEMBL618018

SCHEMBL618018

CCN1CCc2cc(N)ccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATAD2 Q6PL18 1/20 0.55
NOTUM Q6P988 1/20 0.47
MAPT P10636 6/20 0.44
GAA P10253 4/20 0.44
RAD52 P43351 3/20 0.44
GFER P55789 2/20 0.44
HRH3 Q9Y5N1 1/20 0.41
KDM4E B2RXH2 4/20 0.40
S1PR1 P21453 1/20 0.39
ALDH1A1 P00352 6/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
USP2 O75604 1/20 0.39
CDK4 P11802 1/20 0.39
ALOX15 P16050 1/20 0.39
CCND1 P24385 1/20 0.39
ACHE P22303 1/20 0.39
PTK2B Q14289 2/20 0.39
THRB P10828 1/20 0.39
NR4A1 P22736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30168583 1.00 ATAD2 (0.55) ATAD2NOTUMMAPTGAARAD52
SCHEMBL10493943 0.90 ATAD2 (0.53) ATAD2NOTUMMAPTGAARAD52
SCHEMBL3656320 0.86 MAPT (0.49) ATAD2NOTUMMAPTGAARAD52
SCHEMBL2267570 0.86 HTR2A (0.45) ATAD2NOTUMMAPTGAARAD52
Hydrochloric Acid SCHEMBL6844552 0.84 HTR2A (0.44) ATAD2NOTUMMAPTGAARAD52
SCHEMBL24077203 0.81 HTR2A (0.46) ATAD2MAPTGAARAD52GFER
SCHEMBL3437431 0.80 NOTUM (0.51) NOTUMHRH3KDM4EALDH1A1MEN1
SCHEMBL18426670 0.80 ATAD2 (0.43) ATAD2NOTUMMAPTGAARAD52
SCHEMBL4005243 0.80 NOS3 (0.46) ATAD2MAPTGAARAD52GFER
SCHEMBL15068983 0.79 MAPT (0.47) ATAD2MAPTGAARAD52GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357638-A1 MONOAZO DICHROIC DYE COMPOUND, POLARIZING PLATE COMPOSITION COMPRISING SAME, POLARIZING PLATE FORMED THEREFROM, AND OPTICAL DEVICE COMPRISING SAME LG CHEM, LTD. (KR) 2023-11-09 US disclosed
US-20230202989-A1 COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2023-06-29 US disclosed
US-20230202989-A1 COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2023-06-29 US disclosed
WO-2021239885-A1 COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2021-12-02 WO disclosed
EP-3856186-A1 SMALL MOLECULE INHIBITORS OF DYRK1/CLK AND USES THEREOF Arizona Board of Regents on behalf of the University of Arizona (US) 2021-08-04 EP disclosed
WO-2020069418-A1 SMALL MOLECULE INHIBITORS OF DYRK1/CLK AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2020-04-02 WO disclosed
US-20120041207-A1 Compound STERIX LIMITED (GB) 2012-02-16 US disclosed
EP-2293122-A2 Polarizing film, laminate, and liquid crystal display device Fujifilm Corporation (JP) 2011-03-09 EP disclosed
US-20110009448-A1 Compound STERIX LIMITED 2011-01-13 US disclosed
US-7786152-B2 Compound STERIX LIMITED (GB) 2010-08-31 US disclosed
EP-2141163-A1 Substituted thiazolidinones, their production and utilisation as medicine Bayer Schering Pharma AG (DE) 2010-01-06 EP disclosed
US-20080114042-A1 Inhibiting 11 beta-hydroxysteroid dehydrogenase (11 beta-HSD); use of sulfonamide-substituted N-heterocyclics including pyrroles, oxazoles, thiazoles, imidazoles and their fused analogs to treat diabetes, obesity, hypertension, arthritis, asthma, osteoporosis, breast cancer STERIX LIMITED (GB) 2008-05-15 US disclosed
US-7309715-B2 Compound STERIX LIMITED (GB) 2007-12-18 US disclosed
EP-1556040-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 AND TYPE 2 Sterix Limited (GB) 2005-07-27 EP disclosed
US-20040143124-A1 Compound STERIX LIMITED (GB) 2004-07-22 US disclosed
WO-2004037251-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 AND TYPE 2 STERIX LIMITED (GB) 2004-05-06 WO disclosed
EP-1181004-A1 OXIDATION DYEING COMPOSITION FOR KERATINOUS FIBRES AND DYEING METHOD USING SAME L'OREAL (FR) 2002-02-27 EP disclosed
WO-2001066072-A1 OXIDATION DYEING COMPOSITION FOR KERATINOUS FIBRES AND DYEING METHOD USING SAME L'OREAL (FR) 2001-09-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230202989-A1 COMPOUNDS NLRP3, NLRP1, IL1B ATAD2 2496/4885NOTUM 2088/4885MAPT 1004/4885
US-20080114042-A1 Inhibiting 11 beta-hydroxysteroid dehydrogenase (11 beta-HSD); use of sulfonamide-substituted N-heterocyclics including pyrroles, oxazoles, thiazoles, imidazoles and their fused analogs to treat diabetes, obesity, hypertension, arthritis, asthma, osteoporosis, breast cancer HSD11B1, HSD3B1, HSD11B2 ATAD2 3726/4885NOTUM 382/4885MAPT 4759/4885
US-20110009448-A1 Compound NR4A1, GPR6, PRMT6 ATAD2 3805/4885NOTUM 2137/4885MAPT 4794/4885
US-20120041207-A1 Compound NR4A1, GPR6, PRMT6 ATAD2 3805/4885NOTUM 2137/4885MAPT 4794/4885
US-20040143124-A1 Compound NR4A1, CBR1, NR2C2 ATAD2 3996/4885NOTUM 2440/4885MAPT 4691/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.