SCHEMBL29923237

SCHEMBL29923237

CCc1cc(C(=O)O)c2nc(C)ccc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.43
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
GABRA4 P48169 1/20 0.41
GABRE P78334 1/20 0.41
GABRA6 Q16445 1/20 0.41
GABRG1 Q8N1C3 1/20 0.41
GABRG3 Q99928 1/20 0.41
GABRQ Q9UN88 1/20 0.41
SORT1 Q99523 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29924057 0.84 RAB9A (0.42) PARP1RAB9ASORT1NPC1MEN1
SCHEMBL28172844 0.79 PARP1 (0.46) PARP1RAB9ASMN1; SMN2SORT1NPC1
SCHEMBL17035383 0.78 ACLY (0.48) PARP1RAB9ASMN1; SMN2SORT1PKM
SCHEMBL29923343 0.77 PARP1 (0.52) PARP1SMN1; SMN2LMNAALDH1A1KDM4E
SCHEMBL2015530 0.75 KDM4E (0.49) PARP1RAB9ASMN1; SMN2NPC1LMNA
SCHEMBL29923496 0.73 RAB9A (0.43) PARP1RAB9ANPC1MEN1KMT2A
SCHEMBL10947807 0.72 HMGB1 (0.47) RAB9ASMN1; SMN2GABRPGABRDGABRA1
SCHEMBL29412561 0.71 PARP1 (0.72) PARP1RAB9AMEN1KMT2ACCR1
SCHEMBL5319765 0.71 PARP1 (0.72) PARP1RAB9AMEN1KMT2ACCR1
SCHEMBL8072226 0.71 GABRP (0.68) RAB9ASMN1; SMN2GABRPGABRDGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed