SCHEMBL29923449

SCHEMBL29923449

COc1cc(Br)c2nc(C)cc(O)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.41
HPGD P15428 2/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CRHR1 P34998 2/20 0.38
PRNP P04156 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 1/20 0.37
NOD2 Q9HC29 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
MAPT P10636 3/20 0.36
GAA P10253 1/20 0.36
NQO2 P16083 4/20 0.36
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20521814 0.83 CYP3A4 (0.44) CYP3A4HPGDALDH1A1POLBKDM4E
SCHEMBL24915777 0.83 MAPT (0.42) HPGDALDH1A1POLBKDM4EHSD17B10
SCHEMBL20680327 0.78 LMNA (0.38) CYP3A4HPGDALDH1A1KDM4EHSD17B10
SCHEMBL29923651 0.75 L3MBTL1 (0.41) HPGDALDH1A1POLBKDM4EPRNP
SCHEMBL9830239 0.75 NQO2 (0.46) HPGDALDH1A1POLBCRHR1PRNP
SCHEMBL29923598 0.74 HPGD (0.48) CYP3A4HPGDALDH1A1POLBKDM4E
SCHEMBL22750299 0.73 CRHR1 (0.47) CYP3A4ALDH1A1POLBCRHR1PRNP
SCHEMBL29923906 0.73 CRHR1 (0.47) CYP3A4ALDH1A1POLBCRHR1PRNP
SCHEMBL24916103 0.73 NOS3 (0.41) CYP3A4HPGDALDH1A1KDM4ENPSR1
SCHEMBL29924149 0.73 NOS3 (0.41) CYP3A4HPGDALDH1A1KDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed