SCHEMBL29927604

SCHEMBL29927604

NC(=O)c1cccnc1-c1cccc(OCC2COC2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.42
SLC16A3 O15427 3/20 0.42
SLC16A1 P53985 3/20 0.42
MCTS1 Q9ULC4 1/20 0.42
GRM5 P41594 1/20 0.40
PARP10 Q53GL7 3/20 0.40
PARP15 Q460N3 2/20 0.40
PARP1 P09874 3/20 0.39
IGF1R P08069 2/20 0.39
DYRK3 O43781 1/20 0.38
MAP4K4 O95819 1/20 0.38
PIM1 P11309 1/20 0.38
RPS6KB1 P23443 1/20 0.38
CSNK2A1 P68400 1/20 0.38
PKN2 Q16513 1/20 0.38
PIM3 Q86V86 1/20 0.38
BRSK1 Q8TDC3 1/20 0.38
AURKB Q96GD4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6174339 0.80 TTK (0.52) DYRK3MAP4K4PIM1RPS6KB1CSNK2A1
SCHEMBL29927534 0.78 JAK2 (0.37) PARP1DYRK3MAP4K4PIM1RPS6KB1
SCHEMBL6174210 0.77 JAK2 (0.56) PARP1CLK4JAK2
SCHEMBL29927573 0.75 DYRK3 (0.39) SIRT2PARP1DYRK3MAP4K4PIM1
SCHEMBL6174664 0.74 KCNA5 (0.49) GRM5RPS6KB1
SCHEMBL18580116 0.70 TLR8 (0.51) IRAK4PARP1MAP4K4PIM1AURKB
SCHEMBL2991676 0.70 LMNA (0.57) IRAK4PARP1MAP4K4PIM1RPS6KB1
SCHEMBL27964788 0.70 RORB (0.68) PARP1RPS6KB1RORBJAK2
SCHEMBL30108241 0.70 CDC7 (0.53) PARP1CLK4RORB
SCHEMBL945856 0.69 KDM4E (0.55) PARP1CLK4RORBJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022197740-A1 BIARYL AMIDE AND HETEROARYL AMIDES FOR TREATMENT OF CANDIDA ALBICANS INFECTION BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-09-22 WO claimed