SCHEMBL6174664

SCHEMBL6174664

NC(=O)c1cccnc1-c1cccc(OC(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.49
KCNH2 Q12809 1/20 0.49
ROCK2 O75116 1/20 0.49
PDE4A P27815 2/20 0.48
PDE4B Q07343 2/20 0.48
PDE4D Q08499 2/20 0.48
PDE4C Q08493 1/20 0.48
DHODH Q02127 2/20 0.47
DYRK1A Q13627 3/20 0.47
RUNX1 Q01196 1/20 0.47
GSK3B P49841 1/20 0.46
MAPK14 Q16539 1/20 0.46
SLC6A7 Q99884 1/20 0.46
GPR52 Q9Y2T5 1/20 0.44
NPY5R Q15761 1/20 0.44
RPS6KB1 P23443 3/20 0.43
CSNK2A2 P19784 1/20 0.43
CSNK2B P67870 1/20 0.43
CSNK1D P48730 1/20 0.43
CSNK1E P49674 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15391762 0.85 TRPV1 (0.53) ROCK2DHODHRUNX1
SCHEMBL6174210 0.83 JAK2 (0.56) PDE4BDHODHDYRK1A
SCHEMBL6174339 0.81 TTK (0.52) KCNH2PDE4ADHODHRPS6KB1
SCHEMBL5178386 0.80 PARP1 (0.58) KCNA5KCNH2DHODHRPS6KB1
SCHEMBL5518570 0.80 RAB9A (0.56) ROCK2GPR52RPS6KB1
SCHEMBL5498010 0.79 BCAT2 (0.54) DHODHDYRK1A
SCHEMBL2991676 0.78 LMNA (0.57) ROCK2PDE4APDE4BPDE4DPDE4C
SCHEMBL10094730 0.77 KCNH2 (0.54) KCNA5KCNH2PDE4APDE4BPDE4D
SCHEMBL5079789 0.77 LMNA (0.66) KCNH2DHODH
SCHEMBL13387847 0.76 KCNH2 (0.51) KCNA5KCNH2PDE4APDE4BPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575918-A2 SUBSTITUTED BIARYL-4-CARBOXYLIC ACID ARYLAMIDE ANALOGUES AS CAPSAICIN RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2005-09-21 EP claimed
WO-2004056774-A2 SUBSTITUTED BIPHENYL-4-CARBOXYLIC ACID ARYLAMIDE ANALOGUES AS CAPSAICIN RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2004-07-08 WO claimed