SCHEMBL29930730

SCHEMBL29930730

C[Si](C)(C)CCOCn1ncc2cc(-c3cnn(Cc4ccccc4)c3)cnc21

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.45
CREBBP Q92793 5/20 0.43
ALK Q9UM73 1/20 0.41
PIK3CD O00329 2/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41
PI4KA P42356 1/20 0.41
PIK3CG P48736 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
FFAR4 Q5NUL3 1/20 0.39
IKBKE Q14164 2/20 0.38
TBK1 Q9UHD2 2/20 0.38
HDAC8 Q9BY41 1/20 0.37
DHODH Q02127 1/20 0.37
ADORA2A P29274 2/20 0.37
ADORA1 P30542 1/20 0.37
ADORA2B P29275 1/20 0.37
KDM5B Q9UGL1 1/20 0.36
DYRK1B Q9Y463 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29930558 0.77 DYRK1B (0.48) L3MBTL1CREBBPALKPIK3CDPIK3CA
SCHEMBL29930600 0.77 HDAC8 (0.36) CREBBPHDAC8
SCHEMBL29930423 0.76 MAP4K4 (0.40) CREBBP
SCHEMBL29930403 0.76 FTO (0.39) CREBBPPIK3CA
SCHEMBL29930814 0.75 PDGFRB (0.41)
SCHEMBL29930774 0.73 DGAT1 (0.41) CREBBP
SCHEMBL31469272 0.73 DGAT1 (0.35) CREBBP
SCHEMBL19065358 0.73 PIK3CD (0.42) L3MBTL1CREBBPPIK3CDPIK3CAPIK3CB
SCHEMBL31181688 0.73 PIK3CD (0.42) L3MBTL1CREBBPPIK3CDPIK3CAPIK3CB
SCHEMBL31469224 0.73 DGAT1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022235097-A1 PHARMACEUTICAL COMPOSITION CONTAINING NOVEL PYRAZOLO[3,4-B]PYRIDINE DERIVATIVE FOR PREVENTION OR TREATMENT OF METABOLIC DISEASE INCLUDING OBESITY AND DIABETES MELLITUS OR NONALCOHOLIC STEATOHEPATITIS 한국화학연구원 2022-11-10 WO disclosed