SCHEMBL29957280

SCHEMBL29957280

CN(Cc1cc(Br)cs1)c1ccc(C=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.44
CYP2A13 Q16696 1/20 0.44
ALDH1A1 P00352 5/20 0.42
ALDH1A3 P47895 3/20 0.42
ALDH3A1 P30838 3/20 0.42
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
APP P05067 3/20 0.32
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
MEN1 O00255 2/20 0.31
POLB P06746 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2561276 0.80 ALDH1A3 (0.41) CYP2A6CYP2A13ALDH1A1ALDH1A3ALDH3A1
SCHEMBL2561890 0.80 HSP90AA1 (0.36) CYP2A6ALDH1A1HSP90AA1HSP90AB1CYP2C9
SCHEMBL2560536 0.79 ALDH1A3 (0.40) ALDH1A1ALDH1A3ALDH3A1HSP90AA1HSP90AB1
SCHEMBL29952071 0.75 SLC6A4 (0.38) CYP2A6ALDH1A1ALDH1A3HSP90AA1HSP90AB1
SCHEMBL29953414 0.74 GAA (0.50) CYP2A6ALDH1A1HSP90AA1HSP90AB1CYP2C9
SCHEMBL29958389 0.71 RAB9A (0.47) CYP2A6ALDH1A1MAOAMAOBMEN1
SCHEMBL13645995 0.70 CYP2A6 (0.64) CYP2A6CYP2A13ALDH1A1ALDH1A3ALDH3A1
SCHEMBL2514420 0.70 ALDH1A1 (0.65) CYP2A6CYP2A13ALDH1A1ALDH1A3ALDH3A1
SCHEMBL4049989 0.69 CYP2A6 (0.52) CYP2A6CYP2A13ALDH1A1ALDH1A3ALDH3A1
SCHEMBL29953784 0.69 PYCR1 (0.35) ALDH1A1HSP90AA1HSP90AB1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed