SCHEMBL29960848

SCHEMBL29960848

CN(C)CCc1c(N2CCNCC2)ccc(C(N)=O)c1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 3/20 0.39
HTR6 P50406 4/20 0.36
USP28 Q96RU2 1/20 0.34
USP25 Q9UHP3 1/20 0.34
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
ALOX15 P16050 1/20 0.34
GFER P55789 1/20 0.34
YWHAG P61981 1/20 0.34
KMT2A Q03164 1/20 0.34
PARP1 P09874 2/20 0.34
HTT P42858 2/20 0.33
TGFBR1 P36897 1/20 0.33
BRD4 O60885 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30542904 0.99 ACVR1 (0.38) ACVR1HTR6USP28USP25KDM4E
Ammonia Solution, Strong SCHEMBL29115506 0.99 ACVR1 (0.38) ACVR1HTR6USP28USP25KDM4E
SCHEMBL25366356 0.79 HTR6 (0.44) ACVR1HTR6USP28USP25KDM4E
SCHEMBL5666319 0.73 HTR1A (0.47) HTR6HSD17B10PARP1TSHRHTR1A
SCHEMBL30046455 0.71 HTR2C (0.41) HTR6HSD17B10HTTALDH1A1HTR1A
SCHEMBL27675711 0.71 ADRB1 (0.49) ACVR1HTR6KDM4EHSD17B10MEN1
Hydrochloric Acid SCHEMBL31349206 0.70 ADRB1 (0.47) ACVR1HTR6KDM4EHSD17B10MEN1
SCHEMBL30798658 0.70 ACVR1 (0.45) ACVR1MAPTPARP1TGFBR1ALDH1A1
Hydrochloric Acid SCHEMBL27844227 0.70 ADRB1 (0.47) ACVR1HTR6KDM4EHSD17B10MEN1
SCHEMBL9283309 0.69 DRD2 (0.52) HTR6KDM4EHSD17B10PARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222966-A1 SELECTIVE PARP1 INHIBITOR AND APPLICATION THEREOF 成都百裕制药股份有限公司 2022-10-27 WO disclosed