SCHEMBL29968481

SCHEMBL29968481

N#Cc1c(F)cccc1-c1ccc(Br)cn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 2/20 0.38
GABRB3 P28472 2/20 0.38
GABRA5 P31644 2/20 0.38
GABRA3 P34903 2/20 0.38
GABRA1 P14867 1/20 0.38
KDM4E B2RXH2 5/20 0.36
HPGD P15428 4/20 0.36
NPSR1 Q6W5P4 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
BCAT1 P54687 1/20 0.35
ALDH1A1 P00352 4/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPC1 O15118 1/20 0.34
ADORA1 P30542 2/20 0.34
ADORA2A P29274 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28871263 1.00 GABRG2 (0.38) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL2407760 0.79 NPC1 (0.53) HPGDSMN1; SMN2NPC1MEN1KMT2A
SCHEMBL16681034 0.76 SQOR (0.45) KDM4EHPGDALDH1A1GLAGAA
SCHEMBL2147424 0.75 PTGES (0.42) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL28371929 0.74 PTGES (0.52) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL19062287 0.74 ALDH1A1 (0.46) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL6119856 0.74 GRM5 (0.43) KDM4EHPGDALDH1A1GLAGAA
SCHEMBL2650208 0.73 GABRA5 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL17630035 0.73 EGLN2 (0.43) GABRG2GABRB3GABRA5GABRA3ALOX5AP
SCHEMBL28871243 0.72 CASP3 (0.40) GABRG2GABRB3GABRA5GABRA3GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed