SCHEMBL30005327

SCHEMBL30005327

Fc1ccc(OC(F)F)cn1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.39
CHRNA4 P43681 3/20 0.39
DRD1 P21728 1/20 0.37
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HSP90AA1 P07900 1/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
CCR6 P51684 1/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
ALOX15 P16050 1/20 0.36
GFER P55789 1/20 0.36
ADAM17 P78536 1/20 0.36
ROCK1 Q13464 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24665317 1.00 CHRNB2 (0.39) CHRNB2CHRNA4DRD1MEN1ALDH1A1
SCHEMBL31043196 0.81 SYK (0.43) CHRNB2CHRNA4KMT2A
SCHEMBL4741323 0.81 SYK (0.43) CHRNB2CHRNA4KMT2A
SCHEMBL29433330 0.77 CHRNA3 (0.41) CHRNB2CHRNA4LMNAKMT2A
SCHEMBL27978361 0.77 ALOX15 (0.39) DRD1MEN1ALDH1A1LMNAHSP90AA1
SCHEMBL19837604 0.77 DRD1 (0.36) DRD1MEN1ALDH1A1LMNAHSP90AA1
SCHEMBL1002255 0.77 MPO (0.43) DRD1MEN1ALDH1A1LMNAHSP90AA1
SCHEMBL12147787 0.77 RXRA (0.41) CHRNB2CHRNA4DRD1KMT2A
SCHEMBL30187182 0.77 ALOX15 (0.39) CHRNB2CHRNA4DRD1MEN1ALDH1A1
SCHEMBL2895317 0.77 ALOX15 (0.39) CHRNB2CHRNA4DRD1MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4323062-A1 HETEROARYL AMINOPROPANOL DERIVATIVES AS INHIBITORS OF LTA4H Novartis AG (CH) 2024-02-21 EP disclosed
EP-4143194-A1 CD73 INHIBITING 2,4-DIOXOPYRIMIDINE COMPOUNDS GILEAD SCIENCES, INC. (US) 2023-03-08 EP disclosed
WO-2022219546-A1 HETEROARYL AMINOPROPANOL DERIVATIVES AS INHIBITORS OF LTA4H NOVARTIS AG (CH) 2022-10-20 WO disclosed