SCHEMBL1002255

SCHEMBL1002255

Nc1ccc(OC(F)F)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.43
TPO P07202 1/20 0.43
EPX P11678 1/20 0.43
LPO P22079 1/20 0.43
ROCK1 Q13464 1/20 0.41
LTA4H P09960 1/20 0.41
NOS3 P29474 1/20 0.40
NOS2 P35228 1/20 0.40
MBOAT4 Q96T53 1/20 0.39
PDE4A P27815 1/20 0.37
DHFR P00374 1/20 0.36
DRD1 P21728 1/20 0.36
PIK3CD O00329 2/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL22395324 0.98 MPO (0.42) MPOTPOEPXLPOROCK1
SCHEMBL28979546 0.84 MPO (0.41) MPOTPOEPXLPOLTA4H
SCHEMBL1000603 0.81 NOS3 (0.46) MPOTPOEPXLPOLTA4H
Hydrochloric Acid SCHEMBL710140 0.79 NOS3 (0.45) MPOTPOEPXLPOLTA4H
SCHEMBL24665317 0.77 CHRNB2 (0.39) ROCK1DRD1LMNAKMT2AMEN1
SCHEMBL30005327 0.77 CHRNB2 (0.39) ROCK1DRD1LMNAKMT2AMEN1
SCHEMBL30461582 0.76 MPO (0.41) MPOTPOEPXLPOLTA4H
SCHEMBL28663680 0.76 MPO (0.41) MPOTPOEPXLPOLTA4H
SCHEMBL21275802 0.76 ROCK1 (0.41) MPOROCK1MBOAT4DHFRDRD1
SCHEMBL12147787 0.75 RXRA (0.41) MBOAT4DRD1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12384773-B2 Thiazole compounds and methods of use thereof ARCUS BIOSCIENCES, INC. (US) 2025-08-12 US disclosed
WO-2025125665-A1 FURTHER SUBSTITUTED IMIDAZOLES AS INHIBITORS OF NAV1.8 Grünenthal GmbH (DE) 2025-06-19 WO disclosed
US-20250145606-A1 THIAZOLE COMPOUNDS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2025-05-08 US disclosed
WO-2025096979-A1 THIAZOLE COMPOUNDS AS KIT INHIBITORS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2025-05-08 WO disclosed
CN-113754679-B Substituted pyrimidinediones and their use 广东东阳光药业有限公司 2023-04-07 CN disclosed
CN-113754679-A Substituted pyrimidinediones and their use 广东东阳光药业有限公司 2021-12-07 CN disclosed
US-10385012-B2 Thioamides and amides for controlling animal pests BASF SE (DE) 2019-08-20 US disclosed
EP-3049396-B1 PROCESS AND INTERMEDIATES FOR PREPARING INDANYLOXYDIHYDROBENZOFURANYL ACETIC ACID DERIVATIVES AS GPR40 AGONISTS BOEHRINGER INGELHEIM INT (DE) 2017-11-15 EP disclosed
EP-2788086-B1 SUBSTITUTED PYRAZOLES AS MGLU5 RECEPTOR MODULATORS BOEHRINGER INGELHEIM INT (DE) 2016-10-12 EP disclosed
CN-105431420-A Diheteroaryl compounds and uses thereof HOFFMANN LA ROCHE 2016-03-23 CN disclosed
CN-104918934-A 3-substituted pyrazoles and their use as DLK inhibitors HOFFMANN LA ROCHE 2015-09-16 CN disclosed
CN-104352492-A Long-chain fatty acyl elongase inhibitor comprising arylsulfonyl derivative as active ingredient MSD KK 2015-02-18 CN disclosed
EP-2280001-B1 LONG-CHAIN FATTY ACID ELONGATION ENZYME INHIBITOR COMPRISING ARYLSULFONYL DERIVATIVE AS ACTIVE INGREDIENT MSD KK (JP) 2014-10-15 EP disclosed
CN-102015686-B Novel heterocyclic compounds and uses therof NOVARTIS AG 2014-07-02 CN disclosed
US-8420823-B2 Long-chain fatty acyl elongase inhibitor comprising arylsulfonyl derivative as active ingredient MSD K.K. (JP) 2013-04-16 US disclosed
CN-102015638-A Long-chain fatty acid elongase inhibitor containing arylsulfonyl derivative as active ingredient BANYU PHARMA CO LTD 2011-04-13 CN disclosed
EP-2280001-A1 LONG-CHAIN FATTY ACID ELONGATION ENZYME INHIBITOR COMPRISING ARYLSULFONYL DERIVATIVE AS ACTIVE INGREDIENT Banyu Pharmaceutical Co., Ltd. (JP) 2011-02-02 EP disclosed
US-20110009622-A1 LONG-CHAIN FATTY ACYL ELONGASE INHIBITOR COMPRISING ARYLSULFONYL DERIVATIVE AS ACTIVE INGREDIENT MSD K.K. (JP) 2011-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110009622-A1 LONG-CHAIN FATTY ACYL ELONGASE INHIBITOR COMPRISING ARYLSULFONYL DERIVATIVE AS ACTIVE INGREDIENT ELOVL1, ELOVL6, ELOVL3 MPO 2730/4885TPO 3393/4885EPX 452/4885
US-12384773-B2 Thiazole compounds and methods of use thereof TPMT, CYP11B2, ABAT MPO 853/4885TPO 76/4885EPX 258/4885
US-10385012-B2 Thioamides and amides for controlling animal pests TST, TMT1A, ACHE MPO 2445/4885TPO 940/4885EPX 2077/4885
US-20250145606-A1 THIAZOLE COMPOUNDS AND METHODS OF USE THEREOF TPMT, CYP11B2, ABAT MPO 853/4885TPO 76/4885EPX 258/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.