SCHEMBL300143

SCHEMBL300143

[CH2]CC(C)N1CCOCC1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 2/20 0.38
ALDH1A1 P00352 5/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GAA P10253 1/20 0.35
USP2 O75604 1/20 0.33
KCNA5 P22460 1/20 0.33
PKM P14618 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8650528 0.82 KMT2A (0.46) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL1477384 0.81 KMT2A (0.41) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL15174366 0.79 KMT2A (0.44) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL23108665 0.78 KMT2A (0.42) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL21564194 0.78 KMT2A (0.42) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL643674 0.78 KMT2A (0.42) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL10379099 0.77
SCHEMBL23254089 0.76 KMT2A (0.41) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL24245270 0.76 KMT2A (0.41) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL20988251 0.76 KMT2A (0.41) KMT2AMEN1LMNAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 83 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210228525-A1 Methods of Administering Monomethyl Fumarate and Prodrugs Thereof Having Reduced Side Effects ARBOR PHARMACEUTICALS, LLC 2021-07-29 US claimed
US-9302977-B2 Method of making monomethyl fumarate XENOPORT, INC. (US) 2016-04-05 US claimed
EP-2887934-A1 METHODS OF ADMINISTERING MONOMETHYL FUMARATE AND PRODRUGS THEREOF HAVING REDUCED SIDE EFFECTS XenoPort, Inc. (US) 2015-07-01 EP claimed
EP-2854795-A1 TREATMENT OF MULTIPLE SCLEROSIS AND PSORIASIS USING PRODRUGS OF METHYL HYDROGEN FUMARATE XenoPort, Inc. (US) 2015-04-08 EP claimed
WO-2014197860-A1 METHOD OF MAKING MONOMETHYL FUMARATE XENOPORT, INC. (US) 2014-12-11 WO claimed
US-20140364604-A1 METHOD OF MAKING MONOMETHYL FUMARATE HPS INVESTMENT PARTNERS, LLC, AS ADMINISTRATIVE AGENT 2014-12-11 US claimed
US-20140350018-A9 Methods of Administering Monomethyl Fumarate and Prodrugs Thereof Having Reduced Side Effects XENOPORT, INC. (US) 2014-11-27 US claimed
WO-2014031844-A1 METHODS OF ADMINISTERING MONOMETHYL FUMARATE AND PRODRUGS THEREOF HAVING REDUCED SIDE EFFECTS XENOPORT, INC. (US) 2014-02-27 WO claimed
US-20140057917-A1 Methods of Administering Monomethyl Fumarate and Prodrugs Thereof Having Reduced Side Effects XENOPORT, INC. (US) 2014-02-27 US claimed
WO-2013181451-A1 TREATMENT OF MULTIPLE SCLEROSIS AND PSORIASIS USING PRODRUGS OF METHYL HYDROGEN FUMARATE XENOPORT, INC. (US) 2013-12-05 WO claimed
US-20130324539-A1 Treatment of Multiple Sclerosis and Psoriasis Using Prodrugs of Methyl Hydrogen Fumarate WILSHIRE PHARMACEUTICALS, INC. 2013-12-05 US claimed
CN-1203837-C Dye composition containing cationic direct dye and pyraole (1,5-alpha) pyradine as oxidative developing alkali and method of dyeing OREAL (FR) 2005-06-01 CN claimed
CN-1252988-A Dye composition containing cationic direct dye and pyraole (1,5-alpha) pyradine as oxidative developing alkali and method of dyeing OREAL (FR) 2000-05-17 CN claimed
US-20240240229-A1 METHODS OF ADMINISTERING MONOMETHYL FUMARATE AND PRODRUGS THEREOF HAVING REDUCED SIDE EFFECTS HPS INVESTMENT PARTNERS, LLC, AS ADMINISTRATIVE AGENT 2024-07-18 US disclosed
US-20210179573-A1 Treatment of Multiple Sclerosis and Psoriasis Using Prodrugs of Methyl Hydrogen Fumarate ARBOR PHARMACEUTICALS, LLC 2021-06-17 US disclosed
US-20190256480-A1 Treatment of Multiple Sclerosis and Psoriasis Using Prodrugs of Methyl Hydrogen Fumarate ARBOR PHARMACEUTICALS, LLC 2019-08-22 US disclosed
US-5808065-A AMIDATION OF THE CORRESPONDING AMINE COMPOUND TANABE SEIYAKU CO., LTD. (JP) 1998-09-15 US disclosed
US-5378690-A Treatment of angiotensin induced hypertension SANKYO COMPANY, LIMITED (JP) 1995-01-03 US disclosed
EP-0274259-A2 New renin-inhibitory oligopeptides, their preparaton and their use Sankyo Company Limited (JP) 1988-07-13 EP disclosed
US-4686166-A HIGH IMAGE DENSITY, ANTIFOGGING AGENT HITACHI CHEMICAL CO. (JP) 1987-08-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190256480-A1 Treatment of Multiple Sclerosis and Psoriasis Using Prodrugs of Methyl Hydrogen Fumarate MGMT, FH, SI KMT2A 376/4885MEN1 1323/4885LMNA 4823/4885
US-20140057917-A1 Methods of Administering Monomethyl Fumarate and Prodrugs Thereof Having Reduced Side Effects FH, FAH, ALDOA KMT2A 578/4885MEN1 1212/4885LMNA 2857/4885
US-20210179573-A1 Treatment of Multiple Sclerosis and Psoriasis Using Prodrugs of Methyl Hydrogen Fumarate MGMT, FH, SI KMT2A 376/4885MEN1 1323/4885LMNA 4823/4885
US-20140350018-A9 Methods of Administering Monomethyl Fumarate and Prodrugs Thereof Having Reduced Side Effects FH, FAH, ALDOA KMT2A 578/4885MEN1 1212/4885LMNA 2857/4885
US-20240240229-A1 METHODS OF ADMINISTERING MONOMETHYL FUMARATE AND PRODRUGS THEREOF HAVING REDUCED SIDE EFFECTS GSTM1, GSTM2, GSTA1 KMT2A 438/4885MEN1 1620/4885LMNA 4660/4885
US-20140364604-A1 METHOD OF MAKING MONOMETHYL FUMARATE FH, HNMT, FPGS KMT2A 433/4885MEN1 1689/4885LMNA 4040/4885
US-20210228525-A1 Methods of Administering Monomethyl Fumarate and Prodrugs Thereof Having Reduced Side Effects FH, FAH, ALDOA KMT2A 578/4885MEN1 1212/4885LMNA 2857/4885
US-20130324539-A1 Treatment of Multiple Sclerosis and Psoriasis Using Prodrugs of Methyl Hydrogen Fumarate MGMT, FH, SI KMT2A 376/4885MEN1 1323/4885LMNA 4823/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.