SCHEMBL30060872

SCHEMBL30060872

Cn1[nH]c(=O)c2ccc(N)nc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
TP53 P04637 2/20 0.42
ADORA1 P30542 3/20 0.39
ADORA2A P29274 2/20 0.39
PARP1 P09874 1/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
CA5A P35218 1/20 0.35
PDE4A P27815 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
LDHA P00338 1/20 0.32
DAO P14920 1/20 0.31
NPC1 O15118 1/20 0.31
MITF O75030 1/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31425499 0.78 ALDH1A1 (0.44) ADORA1ADORA2APARP1NOS3NOS1
SCHEMBL9037765 0.69 RXFP1 (0.50) KDM4EADORA1ADORA2APDE4ACYP1A2
SCHEMBL18152241 0.69 LDHA (0.58) KDM4ETP53PARP1PDE4ACYP1A2
SCHEMBL11591420 0.67 KDM4E (0.46) KDM4ETP53ADORA1ADORA2APDE4A
SCHEMBL31425543 0.67 DYRK1A (0.39) KDM4EADORA1ADORA2APDE4A
SCHEMBL20323370 0.66 KDM4E (0.36) KDM4ETP53CYP1A2HPGDCYP2C19
SCHEMBL6639554 0.65 MAT2A (0.46) KDM4EADORA1ADORA2APARP1HPGD
SCHEMBL1813535 0.65 MEN1 (0.42) KDM4ETP53CYP1A2CYP2C9HPGD
SCHEMBL16943061 0.64 MCHR1 (0.47)
SCHEMBL12889714 0.63 NOS3 (0.42) KDM4ETP53ADORA1ADORA2ANOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022253252-A1 HETEROCYCLIC COMPOUNDS USEFUL AS HPK1 INHIBITORS SILEXON BIOTECH CO., LTD. (CN) 2022-12-08 WO disclosed