SCHEMBL30091639

SCHEMBL30091639

NC(=O)c1nnc(Cc2cc(F)c(F)c(F)c2)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 1/20 0.36
AURKA O14965 1/20 0.33
RPS6KB1 P23443 1/20 0.33
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
BTK Q06187 2/20 0.32
MAOB P27338 1/20 0.31
RIPK1 Q13546 1/20 0.31
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30091585 0.85 KDM5A (0.41) GPR52AURKARPS6KB1BTKPARP1
SCHEMBL23927492 0.81 ALDH1A1 (0.39)
SCHEMBL30091689 0.81 RPS6KB1 (0.38) GPR52AURKARPS6KB1PARP1
SCHEMBL30091533 0.81 RIPK1 (0.37) CES2CES1RIPK1
SCHEMBL30091705 0.80 MMP13 (0.41) BTKPARP1
SCHEMBL30091570 0.80 GPR52 (0.43) GPR52AURKARPS6KB1
SCHEMBL15964865 0.79 MAOB (0.39) MAOB
SCHEMBL30091702 0.78 MMP2 (0.36)
SCHEMBL30091645 0.77 GPR52 (0.45) GPR52PARP1
SCHEMBL21190099 0.77 KLKB1 (0.34) BTKPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113166116-B Amido bridged heterocyclic compound, and composition and application thereof 北京赛特明强医药科技有限公司 2022-12-27 CN disclosed