SCHEMBL30201287

SCHEMBL30201287

COc1cccc(OC(C)CNC(=N)CNc2cccc(C)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 12/20 0.56
MTNR1B P49286 12/20 0.56
NPC1 O15118 3/20 0.43
RAB9A P51151 2/20 0.41
DRD4 P21917 1/20 0.41
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ACHE P22303 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30201012 0.88 MTNR1B (0.55) MTNR1AMTNR1BNPC1RAB9ASMN1; SMN2
SCHEMBL30200879 0.88 MTNR1A (0.55) MTNR1AMTNR1BNPC1RAB9AALDH1A1
SCHEMBL30201095 0.85 MTNR1A (0.52) MTNR1AMTNR1BALDH1A1SMN1; SMN2GAA
SCHEMBL30201025 0.82 ALDH1A1 (0.44) MTNR1AMTNR1BALDH1A1MAPT
Xylamidine SCHEMBL31307218 0.82 MTNR1A (0.58) MTNR1AMTNR1BALDH1A1ACHE
SCHEMBL30201393 0.78 MTNR1A (0.48) MTNR1AMTNR1B
SCHEMBL30201042 0.78 MTNR1A (0.56) MTNR1AMTNR1BNPC1RAB9AALDH1A1
SCHEMBL30200758 0.77 MTNR1A (0.47) MTNR1AMTNR1BALDH1A1
SCHEMBL30200979 0.77 MTNR1A (0.47) MTNR1AMTNR1BALDH1A1
SCHEMBL30201055 0.77 ALDH1A1 (0.47) MTNR1AMTNR1BRAB9AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023028086-A1 COMBINATIONS OF PERIPHERAL 5-HT2A RECEPTOR ANTAGONISTS AND CENTRAL 5-HT2A RECEPTOR AGONISTS GILGAMESH PHARMACEUTICALS, INC. (US) 2023-03-02 WO disclosed