SCHEMBL30268221

SCHEMBL30268221

O=C1c2ccccc2C(=O)N1c1cc(-c2ccccc2)ccc1O

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.72
ALDH1A1 P00352 3/20 0.52
ALOX5 P09917 1/20 0.48
NR1H3 Q13133 3/20 0.47
ESR2 Q92731 2/20 0.47
ESR1 P03372 2/20 0.47
ACMSD Q8TDX5 2/20 0.46
DHFR P00374 1/20 0.46
HNF4A P41235 1/20 0.46
MCL1 Q07820 1/20 0.46
PIM3 Q86V86 1/20 0.45
HIPK4 Q8NE63 1/20 0.45
SCN2A Q99250 1/20 0.45
HTT P42858 3/20 0.44
HSD17B10 Q99714 2/20 0.44
MEN1 O00255 2/20 0.44
LMNA P02545 2/20 0.44
MAPT P10636 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21857580 0.86 ALDH1A1 (0.71) TYMSALDH1A1HSD17B10MEN1KMT2A
SCHEMBL23752283 0.85 TYMS (1.00) TYMSMEN1LMNAKMT2A
SCHEMBL6005895 0.81 ESR1 (0.62) TYMSNR1H3ESR2ESR1PIM3
SCHEMBL21953468 0.81 EGFR (0.60) TYMSALDH1A1HSD17B10ATMSMN1; SMN2
SCHEMBL30268541 0.81 EGFR (0.60) TYMSALDH1A1HSD17B10ATMSMN1; SMN2
SCHEMBL12733162 0.80 ESR1 (0.51) TYMSALDH1A1NR1H3ESR2ESR1
SCHEMBL19950447 0.78 CYP3A4 (0.61) TYMSALDH1A1NR1H3ESR2ESR1
SCHEMBL27859806 0.77 SCN2A (0.59) TYMSALDH1A1NR1H3SCN2AHTT
SCHEMBL9067222 0.76 MGLL (0.68) TYMSALDH1A1NR1H3HTTHSD17B10
SCHEMBL2150841 0.76 MEN1 (0.55) ALDH1A1NR1H3ESR2ESR1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230047816-A1 PFKFB3 INHIBITORS AND THEIR USES GERO PTE. LTD. (SG) 2023-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230047816-A1 PFKFB3 INHIBITORS AND THEIR USES PFKFB3, PFKFB4, PFKFB1 TYMS 1009/4885ALDH1A1 1943/4885ALOX5 1876/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.