SCHEMBL30337063

SCHEMBL30337063

O=C1CCc2nn(-c3ccccn3)c(O)c2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 4/20 0.40
PDCD1 Q15116 3/20 0.40
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CCNA1 P78396 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CRBN Q96SW2 1/20 0.37
GRM7 Q14831 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA3 P34903 1/20 0.36
HSD17B10 Q99714 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3R2 O00459 1/20 0.35
PIK3CA P42336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15867016 0.80 GABRA1 (0.41) CCNA2CDK2CCNA1SMN1; SMN2ALDH1A1
SCHEMBL29871089 0.80 GABRA1 (0.44) CCNA2CDK2CCNA1SMN1; SMN2ALDH1A1
SCHEMBL4971846 0.80 GABRA1 (0.44) CCNA2CDK2CCNA1SMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL30337257 0.79 GABRA1 (0.43) CCNA2CDK2CCNA1SMN1; SMN2ALDH1A1
SCHEMBL23648620 0.73 PLD1 (0.41) CCNA2CDK2CCNA1SMN1; SMN2ALDH1A1
SCHEMBL29870923 0.73 PLD1 (0.41) CCNA2CDK2CCNA1SMN1; SMN2ALDH1A1
SCHEMBL28818366 0.72 P2RX7 (0.41) SMN1; SMN2ALDH1A1HSD17B10PIK3CDPIK3R2
SCHEMBL23648633 0.71 ALDH1A1 (0.45) ALDH1A1MAPTHSD17B10
SCHEMBL29019285 0.71 ALDH1A1 (0.35) CCNA2CDK2CCNA1SMN1; SMN2ALDH1A1
SCHEMBL23648784 0.71 ALDH1A1 (0.45) CCNA2CDK2CCNA1ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119156379-A Novel pyrazole derivatives 阿普塔生物治疗公司 2024-12-17 CN disclosed
CN-115916766-A Novel pyrazole derivatives 阿普塔生物治疗公司 2023-04-04 CN disclosed