SCHEMBL30337705

SCHEMBL30337705

CC(C)(C)OC(=O)N[C@H]1C[C@H](CO[Si](C)(C)C(C)(C)C)N(C(=O)OC(C)(C)C)C1=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
PRSS1 P07477 1/20 0.33
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
BTK Q06187 1/20 0.31
ALDH1A1 P00352 1/20 0.31
JAK1 P23458 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22118397 0.91 GAA (0.40) GAANFKB1NFKB2RELAF2
SCHEMBL26045071 0.82 TOP2A (0.34) ALDH1A1
SCHEMBL13613731 0.82 TOP2A (0.34) ALDH1A1
SCHEMBL13613732 0.82 TOP2A (0.34) ALDH1A1
SCHEMBL29580011 0.81 FKBP1A (0.31) ALDH1A1
SCHEMBL29580091 0.81 FKBP1A (0.31) ALDH1A1
SCHEMBL958204 0.76 CHRM2 (0.35) KMT2AL3MBTL1ALDH1A1
SCHEMBL625416 0.76 CHRM2 (0.35) KMT2AL3MBTL1ALDH1A1
SCHEMBL211419 0.76 CHRM2 (0.35) KMT2AL3MBTL1ALDH1A1
SCHEMBL21341218 0.76 FPR1 (0.37) GAANFKB1NFKB2RELAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3897833-B1 INHIBITORS OF APOL1 AND METHODS OF USING SAME VERTEX PHARMA (US) 2026-02-04 EP disclosed
US-20250042878-A1 INHIBITORS OF APOL1 AND METHODS OF USING SAME VERTEX PHARMA (US) 2025-02-06 US disclosed
US-12060346-B2 Inhibitors of APOL1 and methods of using same VERTEX PHARMACEUTICALS INCORPORATED (US) 2024-08-13 US disclosed
CN-113453760-B APOL1 inhibitors and methods of use thereof 弗特克斯药品有限公司 2024-05-24 CN disclosed
US-20230271945-A1 INHIBITORS OF APOL1 AND METHODS OF USING SAME VERTEX PHARMACEUTICALS INCORPORATED 2023-08-31 US disclosed
US-11618746-B2 Inhibitors of APOL1 and methods of using same VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-04-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230271945-A1 INHIBITORS OF APOL1 AND METHODS OF USING SAME APOL1, APOB, SAAL1 GAA 533/4885NFKB1 1679/4885NFKB2 1210/4885
US-12060346-B2 Inhibitors of APOL1 and methods of using same APOL1, APOB, SAAL1 GAA 533/4885NFKB1 1679/4885NFKB2 1210/4885
US-20250042878-A1 INHIBITORS OF APOL1 AND METHODS OF USING SAME APOL1, APOB, SAAL1 GAA 533/4885NFKB1 1679/4885NFKB2 1210/4885
US-11618746-B2 Inhibitors of APOL1 and methods of using same APOL1, APOB, NPC1L1 GAA 997/4885NFKB1 1438/4885NFKB2 996/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.