SCHEMBL30367356

SCHEMBL30367356

CC(C)C(=O)N1CCC(c2cc(-c3ccc(N)cc3)c3c(N)noc3c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.42
KIT P10721 6/20 0.40
KDR P35968 6/20 0.40
FLT3 P36888 6/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 3/20 0.38
TLR9 Q9NR96 2/20 0.37
TLR8 Q9NR97 2/20 0.37
ABL1 P00519 1/20 0.37
LCK P06239 1/20 0.37
FYN P06241 1/20 0.37
CSF1R P07333 1/20 0.37
LYN P07948 1/20 0.37
SRC P12931 1/20 0.37
FLT1 P17948 1/20 0.37
FLT4 P35916 1/20 0.37
BLK P51451 1/20 0.37
NAMPT P43490 2/20 0.37
MET P08581 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30367384 0.80 MAPK1 (0.40) DGAT1KITKDRFLT3SMN1; SMN2
SCHEMBL30367399 0.79 TLR9 (0.42) DGAT1MAPK1TLR9TLR8TLR7
SCHEMBL30367296 0.79 MAPK1 (0.39) DGAT1SMN1; SMN2MAPK1TLR9TLR8
Trifluoroacetic Acid SCHEMBL30367156 0.75 DGAT1 (0.44) DGAT1MAPK1PIK3CD
Trifluoroacetic Acid SCHEMBL29052474 0.75 DGAT1 (0.44) DGAT1MAPK1PIK3CD
SCHEMBL30367699 0.73 KDM1A (0.41) DGAT1MAPK1TLR9TLR8NAMPT
SCHEMBL30367527 0.72 MERTK (0.38) KITSMN1; SMN2ALDH1A1MAPK1TLR9
SCHEMBL30367097 0.72 BTK (0.44) SMN1; SMN2TLR9TLR8
SCHEMBL30367867 0.70 KDM4E (0.40) ALDH1A1MAPK1TLR9TLR8NAMPT
SCHEMBL30367001 0.69 DGAT1 (0.39) DGAT1SMN1; SMN2ALDH1A1MAPK1TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023155886-A1 PYRAZOLOPYRIDINE COMPOUNDS AS TAM INHIBITORS SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2023-08-24 WO disclosed
CN-116437918-A Pyrazolopyridine compounds as TAM inhibitors 上海德琪医药科技有限公司 2023-07-14 CN disclosed
WO-2023051464-A1 PYRAZOLOPYRIDINE COMPOUNDS AS TAM INHIBITORS SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2023-04-06 WO disclosed